An antigonadotropin is a drug which suppresses the activity and/or downstream effects of one or both of the gonadotropins, follicle-stimulating hormone...
8 KB (794 words) - 07:50, 29 April 2024
Antiandrogen (section Antigonadotropins)
and antigonadotropins. AR antagonists work by directly blocking the effects of androgens, while androgen synthesis inhibitors and antigonadotropins work...
158 KB (15,084 words) - 00:05, 12 February 2025
Danazol (category Antigonadotropins)
as a weak androgen and anabolic steroid, a weak progestogen, a weak antigonadotropin, a weak steroidogenesis inhibitor, and a functional antiestrogen. Danazol...
47 KB (3,967 words) - 14:58, 12 January 2025
Gestrinone (category Antigonadotropins)
and antiprogestogen, a weak androgen and anabolic steroid, a weak antigonadotropin, a weak steroidogenesis inhibitor, and a functional antiestrogen. Gestrinone...
27 KB (2,261 words) - 06:20, 14 January 2025
diet or quack preparations, which are illegal in various countries. Antigonadotropin Gonadotropin surge-attenuating factor Parhar, Ishwar S. (2002)....
11 KB (1,114 words) - 23:42, 22 March 2025
precursor of cyproterone acetate (CPA), an antiandrogen, progestin, and antigonadotropin which was introduced instead of cyproterone and is widely used as a...
23 KB (2,367 words) - 08:43, 8 September 2024
Paroxypropione (category Antigonadotropins)
synthetic nonsteroidal estrogen which has been used medically as an antigonadotropin in Spain and Italy but appears to no longer be marketed. It was first...
10 KB (862 words) - 02:30, 8 August 2024
Steroidal antiandrogen (category Antigonadotropins)
Cyproterone acetate (Androcur): A combined AR antagonist and progestogen/antigonadotropin. Also has weak glucocorticoid activity. Previously used widely in the...
24 KB (2,340 words) - 21:47, 24 November 2024
List of antiandrogens (section Antigonadotropins)
inhibitors like 5α-reductase inhibitors and CYP17A1 inhibitors, and antigonadotropins like GnRH analogues, estrogens, and progestogens. In addition, it...
5 KB (254 words) - 18:23, 18 September 2023
Desogestrel (category Antigonadotropins)
In addition, desogestrel has been extensively investigated as an antigonadotropin at dosages of 150 to 300 μg/day in combination with testosterone in...
63 KB (5,560 words) - 14:13, 9 April 2025
testosterone levels; antiandrogens such as androgen receptor antagonists, antigonadotropins, GnRH modulators, and 5α-reductase inhibitors to further oppose the...
231 KB (25,328 words) - 15:03, 9 April 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
25 KB (2,033 words) - 10:47, 9 April 2025
(SERD) fulvestrant, aromatase inhibitors (AIs) like anastrozole, and antigonadotropins including androgens/anabolic steroids, progestogens, and GnRH analogues...
8 KB (745 words) - 20:56, 24 November 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
150 KB (15,796 words) - 14:35, 17 April 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
50 KB (4,376 words) - 16:04, 12 January 2025
steroids. Steroidogenesis inhibitors are analogous in effect and use to antigonadotropins (which specifically inhibit gonadal sex steroid production), but work...
37 KB (2,107 words) - 21:47, 24 November 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
49 KB (4,706 words) - 07:47, 7 April 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
182 KB (17,424 words) - 17:12, 17 April 2025
Gonadotropin-releasing hormone agonist (category Antigonadotropins)
used as a progonadotropin, all approved GnRH agonists are used as antigonadotropins. The clinically used desensitizing GnRH agonists are available in...
26 KB (2,683 words) - 16:35, 15 February 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
23 KB (2,061 words) - 06:21, 14 January 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
209 KB (21,556 words) - 01:54, 21 February 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
70 KB (7,199 words) - 05:12, 11 April 2025
Fadrozole Formestane Third-generation: Anastrozole Exemestane Letrozole Antigonadotropins Androgens/anabolic steroids (e.g., testosterone, testosterone esters...
28 KB (2,348 words) - 22:32, 16 February 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
27 KB (2,353 words) - 02:49, 5 April 2025
of administration Implant Drug class GnRH analogue; GnRH agonist; Antigonadotropin ATC code L02AE03 (WHO) Legal status Legal status CA: ℞-only In general:...
11 KB (820 words) - 13:18, 27 January 2025
inhibits androgen production in the body (i.e., it does not act as an antigonadotropin or androgen steroidogenesis inhibitor or lower androgen levels) and...
221 KB (21,804 words) - 17:52, 16 April 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
18 KB (1,725 words) - 23:33, 17 March 2025
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
48 KB (4,589 words) - 06:41, 7 April 2025
Fadrozole Formestane Third-generation: Anastrozole Exemestane Letrozole Antigonadotropins Androgens/anabolic steroids (e.g., testosterone, testosterone esters...
21 KB (2,055 words) - 21:12, 21 November 2024
Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins D2 receptor antagonists (prolactin releasers) (e.g., domperidone,...
95 KB (9,427 words) - 03:08, 14 April 2025