Conolidine is an indole alkaloid. Preliminary reports suggest that it could provide analgesic effects with few of the detrimental side-effects associated...
10 KB (962 words) - 22:42, 28 August 2024
The species is known to produce many alkaloids including catharanthine, conolidine, coronaridine, dregamine, ibogamine, tabersonine, voacangine, voacamine...
6 KB (490 words) - 15:22, 13 June 2024
naturally occurring alkaloid conolidine. RTI-5152-12 has 15-fold improved potency towards ACKR3 relative to conolidine. ACKR3 is a novel opioid receptor...
10 KB (930 words) - 21:55, 23 September 2024
the genus is known to contain ibogaine (e.g. in bëcchëte, T. undulata), conolidine (present in minor concentration in T. divaricata) and voacangine (T. alba...
15 KB (1,198 words) - 04:47, 9 December 2023
and desomorphine use in North America is still considered unconfirmed. Conolidine Xylazine, a drug with similar side effects, widespread in the United States...
24 KB (2,505 words) - 22:24, 27 September 2024
for instance their analgesic effects. Other ligands of ACKR3 include conolidine, CCX771, RTI-5152-12, and VUF15485. Palmer CB, Meyrath M, Canals M, Kostenis...
9 KB (704 words) - 21:32, 3 September 2024
sensitivity and specificity of the mu-conotoxins for the different isoforms. Conolidine Contryphan, members of "conotoxin O2" Conantokins, also known as "conotoxin...
14 KB (1,477 words) - 19:20, 22 August 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
97 KB (11,021 words) - 17:45, 18 September 2024
including Tabernaemontana divaricata, and in Ervatamia peduncularis. Conolidine Conopharyngine US 20070232533, "Use of Vinca Alkaloids and Salts Thereof" ...
2 KB (77 words) - 18:09, 20 June 2022
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
30 KB (2,931 words) - 15:04, 1 October 2024
inhibitor and butyrylcholinesterase inhibitor isolated from Tabernaemontana. Conolidine Confoline Vieira, IJ; Medeiros, WL; Monnerat, CS; Souza, JJ; Mathias,...
3 KB (113 words) - 23:53, 8 August 2022
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
10 KB (1,231 words) - 22:00, 8 March 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
20 KB (2,419 words) - 23:03, 5 September 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
22 KB (2,786 words) - 02:02, 19 August 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
67 KB (7,852 words) - 18:22, 10 September 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
21 KB (2,612 words) - 11:46, 29 July 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
14 KB (1,641 words) - 23:08, 5 September 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
12 KB (954 words) - 13:32, 23 April 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
20 KB (2,508 words) - 19:36, 5 September 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
14 KB (957 words) - 14:32, 14 June 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
9 KB (885 words) - 07:16, 30 April 2024
g/mol, exact mass: 266.1419 u) may refer to: 5-Benzyloxytryptamine (5-BT) Conolidine Ervaticine This set index page lists chemical structure articles associated...
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CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
3 KB (138 words) - 07:01, 2 December 2023
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
4 KB (518 words) - 21:19, 21 November 2023
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
28 KB (3,148 words) - 11:43, 29 July 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
17 KB (2,039 words) - 03:19, 24 August 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
5 KB (642 words) - 21:49, 2 September 2023
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
4 KB (283 words) - 23:37, 3 December 2023
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
26 KB (2,934 words) - 23:08, 5 September 2024
CXCR4) CXCR5 Agonists: CXCL13 CXCR6 Agonists: CXCL16 CXCR7 Agonists: Conolidine CXCL11 (I-TAC) CCX771 LIH383 RTI-5152-12 SDF-1 (CXCL12) VUF15485 PAMs:...
11 KB (1,456 words) - 17:37, 5 September 2024