H2 receptors are a type of histamine receptor found in many parts of the anatomy of humans and other animals. They are positively coupled to adenylate...
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of histamine at the histamine H2 receptors of the parietal cells in the stomach. This decreases the production of stomach acid. H2 antagonists can be used...
20 KB (2,234 words) - 18:27, 20 October 2024
Antihistamine (redirect from Histamine receptor antagonist)
antihistamines are H1-antihistamines and H2-antihistamines. H1-antihistamines work by binding to histamine H1 receptors in mast cells, smooth muscle, and endothelium...
36 KB (3,292 words) - 00:41, 26 October 2024
bind with histamine, a neurotransmitter involved in various physiological processes. There are four main types: H1, H2, H3, and H4. H1 receptors are linked...
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its receptor. Antihistamine – Histamine receptor antagonists H1-receptor antagonist Histamine H2-receptor Histamine H3-receptor Histamine H4-receptor GRCh38:...
15 KB (1,740 words) - 16:17, 21 August 2024
noradrenaline, histamine and serotonin. The gene sequence for H3 receptors expresses only about 22% and 20% homology with both H1 and H2 receptors respectively...
21 KB (2,345 words) - 06:57, 24 September 2024
during treatment with histamine H2 receptor antagonists such as cimetidine, ranitidine, and risperidone. The injection of histamine into the corpus cavernosum...
50 KB (4,980 words) - 14:10, 25 September 2024
The histamine H4 receptor, like the other three histamine receptors, is a member of the G protein-coupled receptor superfamily that in humans is encoded...
11 KB (1,253 words) - 06:58, 21 July 2024
Famotidine (redirect from H2 Bloc)
Famotidine, sold under the brand name Pepcid among others, is a histamine H2 receptor antagonist medication that decreases stomach acid production. It...
27 KB (2,336 words) - 22:40, 9 November 2024
Cimetidine (category H2 receptor antagonists)
Cimetidine, sold under the brand name Tagamet among others, is a histamine H2 receptor antagonist that inhibits stomach acid production. It is mainly used...
50 KB (5,133 words) - 06:08, 31 October 2024
in the British National Vegetation Classification system Histamine H2 receptor Prostaglandin H2 H-2, the Major histocompatibility complex of the mouse (equivalent...
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Betazole (also known as ametazole) is a histamine H2 receptor agonist. Betazole hydrochloride is known as gastramine and histalog. It has been used as...
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A histamine agonist is a drug which causes increased activity at one or more of the four histamine receptor subtypes. H1 agonists promote wakefulness...
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Hives (section Dietary histamine poisoning)
Fedorowicz, Zbys; van Zuuren, Esther J; Hu, Nianfang (14 March 2012). "Histamine H2-receptor antagonists for urticaria". Cochrane Database of Systematic Reviews...
50 KB (5,769 words) - 14:49, 25 October 2024
Nizatidine (category H2 receptor antagonists)
Nizatidine is a histamine H2 receptor antagonist that inhibits stomach acid production, and is commonly used in the treatment of peptic ulcer disease...
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Lafutidine (category H2 receptor antagonists)
Lafutidine (INN) is a second generation histamine H2 receptor antagonist having multimodal mechanism of action and used to treat gastrointestinal disorders...
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Ranitidine (redirect from Alter-H2)
Clostridioides difficile colitis. Ranitidine is an H2 histamine receptor antagonist that works by blocking histamine, thus decreasing the amount of acid released...
100 KB (8,778 words) - 03:03, 23 October 2024
Metiamide (category H2 receptor antagonists)
Metiamide is a histamine H2 receptor antagonist developed from another H2 antagonist, burimamide. It was an intermediate compound in the development of...
6 KB (518 words) - 06:43, 5 January 2024
An H3 receptor antagonist is a type of antihistaminic drug used to block the action of histamine at H3 receptors. Unlike the H1 and H2 receptors which...
19 KB (2,154 words) - 12:44, 26 September 2024
proteins C3a and C5a, bind to receptors on mast cells and basophils causing degranulation. Granules in these cells contain histamine, platelet-activating factor...
44 KB (4,096 words) - 22:53, 25 October 2024
Burimamide (category H2 receptor antagonists)
Burimamide is an antagonist at the H2 and H3 histamine receptors. At physiological pH, it is largely inactive as an H2 antagonist, but its H3 affinity is...
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H1 antagonist (redirect from Histamine h1 antagonists)
blockers, are a class of medications that block the action of histamine at the H1 receptor, helping to relieve allergic reactions. Agents where the main...
23 KB (1,879 words) - 02:48, 28 October 2024
highly potent and specific histamine H2 receptor agonist. It has been used diagnostically as a gastric secretion indicator. Histamine agonists Durant G, Duncan...
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Amthamine (category Histamine agonists)
as other functions of the H2 receptor. Eriks, J. C; Van Der Goot, H; Sterk, G. J; Timmerman, H (1992). "Histamine H2-receptor agonists. Synthesis, in vitro...
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this can lead to higher concentrations of metformin in the body. Histamine H2 receptor antagonists like cimetidine and ranitidine may reduce the efficacy...
25 KB (2,008 words) - 08:23, 19 October 2024
for the histamine H2 receptor, 964 nM for the alpha-2A adrenergic receptor, 115 nM for the serotonin transporter, 4519 nM for the σ1 receptor, and 525...
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MRI or somatostatin receptor scintigraphy. Proton pump inhibitors (such as omeprazole and lansoprazole) and histamine H2-receptor antagonists (such as...
12 KB (1,126 words) - 15:14, 26 October 2024
(TAAR9, TAR3) Histamine H2 receptor (HRH2, HH2R) InterPro: IPR000503 Histamine H1 receptor (HRH1, HH1R) InterPro: IPR000921 Histamine H3 receptor (HRH3) InterPro: IPR003980...
25 KB (2,172 words) - 01:01, 29 November 2023
Zolantidine (category H2 receptor antagonists)
Zolantidine is a brain-penetrating selective histamine H2 receptor (HRH2) antagonist developed by Smith, Kline & French, with the research code of SK&F...
2 KB (98 words) - 16:18, 24 January 2023
A study from 2019 showed that PPI use alone and together with histamine H2-receptor antagonists was associated with an increased bone fracture hazard...
58 KB (6,306 words) - 03:11, 9 November 2024