muscarinic acetylcholine receptor, also known as cholinergic/acetylcholine receptor M3, or the muscarinic 3, is a muscarinic acetylcholine receptor encoded...
16 KB (1,761 words) - 05:18, 24 October 2024
The muscarinic acetylcholine receptor M1, also known as the cholinergic receptor, muscarinic 1, is a muscarinic receptor that in humans is encoded by the...
22 KB (2,227 words) - 08:51, 26 October 2024
The muscarinic acetylcholine receptor M2, also known as the cholinergic receptor, muscarinic 2, is a muscarinic acetylcholine receptor that in humans is...
19 KB (2,091 words) - 17:29, 25 September 2024
The muscarinic acetylcholine receptor M4, also known as the cholinergic receptor, muscarinic 4 (CHRM4), is a protein that, in humans, is encoded by the...
20 KB (2,130 words) - 04:59, 2 December 2024
Muscarinic acetylcholine receptors (mAChRs) are acetylcholine receptors that form G protein-coupled receptor complexes in the cell membranes of certain...
36 KB (3,151 words) - 04:36, 9 December 2024
The human muscarinic acetylcholine receptor M5, encoded by the CHRM5 gene, is a member of the G protein-coupled receptor superfamily of integral membrane...
13 KB (1,511 words) - 04:39, 20 October 2024
proliferative signals via a membrane-located M1-muscarinic receptor homolog. Partly because of acetylcholine's muscle-activating function, but also because...
41 KB (4,382 words) - 05:15, 9 November 2024
"ionotropic" acetylcholine receptors) are particularly responsive to nicotine. The nicotine ACh receptor is also a Na+, K+ and Ca2+ ion channel. Muscarinic acetylcholine...
13 KB (1,309 words) - 04:20, 6 December 2024
A muscarinic acetylcholine receptor agonist, also simply known as a muscarinic agonist or as a muscarinic agent, is an agent that activates the activity...
9 KB (858 words) - 23:25, 21 November 2024
A muscarinic acetylcholine receptor antagonist, also simply known as a muscarinic antagonist or as an antimuscarinic agent, is a type of anticholinergic...
41 KB (2,060 words) - 02:02, 24 November 2024
System Messier 3 (M3), a globular cluster in the constellation Canes Venatici Muscarinic acetylcholine receptor M3, an acetylcholine receptor The M-3 (My Mood...
7 KB (1,017 words) - 18:02, 21 October 2024
Parasympathomimetic drug (redirect from Acetylcholine receptor agonist)
or muscarinic receptors. Choline esters Acetylcholine (all acetylcholine receptors) Bethanechol (M3 receptors) Carbachol (all muscarinic receptors and...
7 KB (618 words) - 06:38, 29 April 2024
Xanomeline (category M3 receptor agonists)
proposed brand names Lumeron, Memcor) is a small molecule muscarinic acetylcholine receptor agonist that was first synthesized in a collaboration between...
22 KB (1,772 words) - 23:58, 9 December 2024
parasympathetic postganglionic fibers releasing acetylcholine acting primarily on the muscarinic acetylcholine receptor (M3) of iris sphincter muscle. Preganglionic...
5 KB (472 words) - 19:22, 14 September 2024
releasing factor type 1 receptor Sphingosine-1-phosphate receptors EDG1, EDG3 and EDG5 Muscarinic acetylcholine receptor M3 Transient receptor potential TRPC1...
25 KB (3,066 words) - 13:23, 9 November 2024
Xanomeline/trospium chloride (category M3 receptor antagonists)
xanomeline, a muscarinic agonist; and trospium chloride, a muscarinic antagonist. Xanomeline is a functionally preferring muscarinic M4 and M1 receptor agonist...
18 KB (1,561 words) - 07:10, 16 November 2024
Sympathetic nervous system Acetylcholine Choline Cholinergic receptor Nicotinic acetylcholine receptor Muscarinic acetylcholine receptor Langley, John Newport...
31 KB (3,865 words) - 01:13, 16 December 2024
Bethanechol (category M3 receptor agonists)
carbamate that selectively stimulates muscarinic receptors without any effect on nicotinic receptors. Unlike acetylcholine, bethanechol is not hydrolyzed by...
7 KB (390 words) - 06:52, 25 October 2024
Desmethylclozapine (category M3 receptor agonists)
muscarinic acetylcholine M1 receptor and the δ-opioid receptor, unlike clozapine as well. It is a moderate-efficacy partial agonist of the muscarinic...
7 KB (639 words) - 23:57, 14 November 2024
Trospium chloride (category M3 receptor antagonists)
affinity for all five of the muscarinic acetylcholine receptor subtypes, including the M1, M2, M3, M4, and M5 receptors. After oral administration, less...
22 KB (2,087 words) - 06:58, 12 November 2024
Cyclobenzaprine (category M3 receptor antagonists)
receptor antagonism. In terms of its antimuscarinic activity, it is said to be an antagonist of the muscarinic acetylcholine M1, M2, and M3 receptors...
31 KB (2,429 words) - 04:38, 5 December 2024
Muscarine (category M3 receptor agonists)
concentrations up to 1.6%. Muscarine is a selective agonist of the muscarinic acetylcholine receptors. The name muscarine derives from that of Amanita muscaria...
18 KB (1,882 words) - 06:42, 25 October 2024
adrenergic receptor kinase Beta adrenergic receptor kinase-2 Acetylcholine receptor (Cholinergic receptor) Nicotinic acetylcholine receptor Muscarinic acetylcholine...
33 KB (2,982 words) - 15:21, 27 November 2024
Methacholine (category M3 receptor agonists)
acetyl-β-methylcholine, is a synthetic choline ester that acts as a non-selective muscarinic receptor agonist in the parasympathetic nervous system. Methacholine is primarily...
6 KB (383 words) - 04:14, 26 October 2024
Benzatropine (category M3 receptor antagonists)
specifically an antimuscarinic and acts a selective muscarinic acetylcholine M1 and M3 receptor antagonist. Benzatropine partially blocks cholinergic...
18 KB (1,439 words) - 07:13, 18 December 2024
Scopolamine (category M3 receptor antagonists)
central muscarinic acetylcholine receptors. Scopolamine acts as a nonspecific muscarinic antagonist at all four (M1, M2, M3, and M4) receptor sites. In...
59 KB (5,256 words) - 20:55, 27 November 2024
Oxotremorine (category M3 receptor agonists)
Oxotremorine is a drug that acts as a selective muscarinic acetylcholine receptor agonist. Oxotremorine produces ataxia, tremor and spasticity, similar...
3 KB (155 words) - 04:14, 26 October 2024
Dicycloverine (category M3 receptor antagonists)
Dicycloverine is a selective muscarinic acetylcholine M1 receptor antagonist. It blocks the action of acetylcholine on muscarinic receptors on smooth muscles in...
13 KB (1,090 words) - 02:18, 25 November 2024
Talsaclidine (category M3 receptor agonists)
non-selective muscarinic acetylcholine receptor agonist which acts as a full agonist at the M1 subtype, and as a partial agonist at the M2 and M3 subtypes...
4 KB (297 words) - 05:39, 26 October 2024
ligands have unique receptors. Some examples include: metabotropic glutamate receptors, muscarinic acetylcholine receptors, GABAB receptors. The G protein-coupled...
6 KB (625 words) - 00:59, 6 June 2024