Gabapentinoids, also known as α2δ ligands, are a class of drugs that are derivatives of the inhibitory neurotransmitter gamma-Aminobutyric acid (GABA)...
41 KB (4,035 words) - 10:47, 19 May 2024
DS-5565) is a gabapentinoid medication developed by Daiichi Sankyo. Gabapentin and pregabalin are also members of this class. As a gabapentinoid, mirogabalin...
5 KB (299 words) - 19:44, 24 October 2023
use in epilepsy is as an add-on therapy for partial seizures. It is a gabapentinoid medication (GABA analogue) which are drugs that are derivatives of γ-aminobutyric...
99 KB (8,532 words) - 22:10, 15 October 2024
the symptoms of opiate withdrawal, there is increasing evidence that gabapentinoids are effective in controlling some of the symptoms during opiate detoxification...
91 KB (8,927 words) - 16:51, 8 October 2024
Depressant (section Gabapentinoids)
include drugs like Xanax (a benzodiazepine) and a number of opioids. Gabapentinoids like gabapentin and pregabalin are depressants and have anticonvulsant...
130 KB (13,432 words) - 06:24, 11 September 2024
Retrieved February 13, 2013. "Review finds little evidence to support gabapentinoid use in bipolar disorder or insomnia". NIHR Evidence (Plain English summary)...
157 KB (17,676 words) - 17:54, 18 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
181 KB (19,613 words) - 04:19, 10 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
95 KB (9,778 words) - 12:09, 15 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
165 KB (15,851 words) - 21:46, 14 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
224 KB (25,904 words) - 22:32, 18 October 2024
subunit-containing VDCCs, similarly to gabapentin and pregabalin, and hence is a gabapentinoid. Both (R)-phenibut and (S)-phenibut display this action with similar...
36 KB (2,964 words) - 16:40, 10 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
103 KB (10,986 words) - 06:41, 16 September 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
159 KB (16,664 words) - 03:57, 9 October 2024
Loperamide Mibefradil NP078585 Ruthenium red TROX-1 α2δ subunit-selective (gabapentinoids): 4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen...
116 KB (11,202 words) - 06:03, 17 October 2024
Regnite (in Japan)) is an anticonvulsant and analgesic drug of the gabapentinoid class, and a prodrug to gabapentin. It was designed for increased oral...
8 KB (648 words) - 21:39, 20 December 2023
GABA-T inhibitor Bamaluzole Bicuculline Deramciclane Ethanol Fengabine Gabapentinoid Loreclezole Propofol Retigabine/ezogabine Tiagabine Valerenic acid John...
8 KB (754 words) - 04:40, 27 January 2024
include: Analgesic Benzodiazepine Cannabinoid Cardiac glycoside Fibrate Gabapentinoid Steroid Thiazide diuretic Triptan β-lactam antibiotic This type of categorisation...
10 KB (1,021 words) - 12:27, 19 August 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
87 KB (8,227 words) - 03:57, 9 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
165 KB (17,242 words) - 10:41, 9 October 2024
Anticonvulsant (section Gabapentinoids)
Vigabatrin and progabide are also analogs of GABA. Topiramate (1995). Gabapentinoids are used in epilepsy, neuropathic pain, fibromyalgia, restless leg syndrome...
70 KB (5,714 words) - 11:37, 30 September 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
142 KB (15,105 words) - 07:45, 29 September 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
156 KB (15,356 words) - 20:21, 18 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
168 KB (16,897 words) - 00:31, 20 October 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
123 KB (12,215 words) - 00:57, 20 October 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
88 KB (7,952 words) - 16:30, 19 October 2024
Loperamide Mibefradil NP078585 Ruthenium red TROX-1 α2δ subunit-selective (gabapentinoids): 4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen...
69 KB (7,678 words) - 03:57, 24 September 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
51 KB (4,614 words) - 05:58, 14 October 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
44 KB (4,711 words) - 18:17, 24 September 2024
Benzodiazepines Carbamates Ethanol (alcohol) Alcoholic beverage Beer Wine Gabapentinoids GHB Inhalants Medical Nitrous oxide (recreational use) Hazardous solvents...
149 KB (13,773 words) - 13:34, 14 October 2024
Carisoprodol Chlormezanone‡ Ethanol (alcohol) Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin...
58 KB (5,390 words) - 03:24, 10 October 2024