• Thumbnail for Nonsteroidal antiandrogen
    A nonsteroidal antiandrogen (NSAA) is an antiandrogen with a nonsteroidal chemical structure. They are typically selective and full or silent antagonists...
    17 KB (1,576 words) - 15:57, 24 February 2024
  • Thumbnail for Antiandrogen
    steroidal antiandrogen that has been widely used in the treatment of prostate cancer, but it has largely been replaced by nonsteroidal antiandrogens, which...
    159 KB (15,079 words) - 15:42, 24 September 2024
  • testosterone levels to the female/castrate range. Nonsteroidal antiandrogens are antiandrogens which are nonsteroidal and hence unrelated to steroid hormones in...
    232 KB (25,231 words) - 16:06, 1 October 2024
  • Thumbnail for List of antiandrogens
    progestogens. In addition, it includes both steroidal antiandrogen (SAAs) and nonsteroidal antiandrogen (NSAAs). 17α-Hydroxyprogesterone derivatives Chlormadinone...
    5 KB (254 words) - 18:23, 18 September 2023
  • Thumbnail for Enzalutamide
    Enzalutamide (category Nonsteroidal antiandrogens)
    Enzalutamide, sold under the brand name Xtandi, is a nonsteroidal antiandrogen (NSAA) medication which is used in the treatment of prostate cancer. It...
    50 KB (4,674 words) - 20:52, 20 August 2024
  • Comparison of the nonsteroidal antiandrogen (NSAA) bicalutamide with other antiandrogens reveals differences between the medications in terms of efficacy...
    85 KB (8,727 words) - 01:24, 2 September 2024
  • (SGRMTooltip Selective glucocorticoid receptor modulator) Nonsteroidal antiandrogen Nonsteroidal estrogen Edward J. Pavlik (6 December 2012). Estrogens,...
    5 KB (381 words) - 23:18, 21 July 2023
  • Thumbnail for Steroidal antiandrogen
    for the same purpose. They are the converse of nonsteroidal antiandrogens (NSAAs), which are antiandrogens that are not steroids and are structurally unrelated...
    24 KB (2,340 words) - 08:04, 7 February 2024
  • Thumbnail for Gynecomastia
    4103/2230-8210.113770. PMC 3743379. PMID 23961495. Gillatt, David (August 2006). "Antiandrogen treatments in locally advanced prostate cancer: are they all the same...
    63 KB (6,551 words) - 04:35, 6 October 2024
  • Thumbnail for Thalidomide
    Thalidomide (category Nonsteroidal antiandrogens)
    acts as an antagonist of the androgen receptor and hence is a nonsteroidal antiandrogen of some capacity. In accordance, it can produce gynecomastia and...
    76 KB (7,430 words) - 22:51, 2 October 2024
  • Thumbnail for Apalutamide
    Apalutamide (category Nonsteroidal antiandrogens)
    Apalutamide, sold under the brand name Erleada among others, is a nonsteroidal antiandrogen (NSAA) medication used for the treatment of prostate cancer. It...
    36 KB (3,026 words) - 22:35, 16 August 2024
  • antiandrogens can potentially be used to treat it. As of 2010[update] antiandrogens are small molecules and can be either steroidal or nonsteroidal depending...
    42 KB (4,594 words) - 12:34, 28 September 2024
  • Thumbnail for Topilutamide
    Topilutamide (category Nonsteroidal antiandrogens)
    known as perfluoroacylamido-arylpropanamides. Topilutamide is a nonsteroidal antiandrogen (NSAA), or an antagonist of the androgen receptor (AR), the biological...
    10 KB (762 words) - 22:08, 3 February 2024
  • Thumbnail for Valproate
    Valproate (category Nonsteroidal antiandrogens)
    antagonist of the androgen and progesterone receptors, and hence as a nonsteroidal antiandrogen and antiprogestogen, at concentrations much lower than therapeutic...
    93 KB (8,024 words) - 20:00, 24 September 2024
  • Thumbnail for Andarine
    osteoporosis, and benign prostatic hypertrophy (BPH), using the nonsteroidal antiandrogen bicalutamide as a lead compound. Development of andarine for all...
    10 KB (958 words) - 17:14, 4 July 2024
  • Thumbnail for Enobosarm
    structural modification of the arylpropionamide nonsteroidal antiandrogen bicalutamide. They are nonsteroidal arylpropionamides themselves and are close structural...
    116 KB (12,935 words) - 04:43, 18 August 2024
  • The medical uses of bicalutamide, a nonsteroidal antiandrogen (NSAA), include the treatment of androgen-dependent conditions and hormone therapy to block...
    134 KB (13,465 words) - 04:59, 3 September 2024
  • Thumbnail for DIMP (antiandrogen)
    7-8117), or N-(3,5-dimethyl-4-isoxazolylmethyl)phthalimide, is a nonsteroidal antiandrogen (NSAA) structurally related to thalidomide (which also binds to...
    7 KB (554 words) - 13:19, 2 March 2024
  • Thumbnail for Spironolactone
    Spironolactone (category Steroidal antiandrogens)
    Spironolactone, the 5α-reductase inhibitor finasteride, and the nonsteroidal antiandrogen flutamide all appear to have similar effectiveness in the treatment...
    181 KB (17,316 words) - 05:17, 7 September 2024
  • Thumbnail for Nilutamide
    Nilutamide (category Nonsteroidal antiandrogens)
    Nilutamide, sold under the brand names Nilandron and Anandron, is a nonsteroidal antiandrogen (NSAA) which is used in the treatment of prostate cancer. It has...
    52 KB (5,386 words) - 16:26, 15 September 2024
  • Thumbnail for RU-58841
    RU-58841 (category Nonsteroidal antiandrogens)
    RU-58841, also known as PSK-3841 or HMR-3841, is a nonsteroidal antiandrogen (NSAA) which was initially developed in the 1980s by Roussel Uclaf, the French...
    6 KB (533 words) - 18:51, 25 October 2023
  • Thumbnail for Pharmacology of bicalutamide
    of the pharmacodynamic and pharmacokinetic properties of the nonsteroidal antiandrogen (NSAA) bicalutamide. In terms of pharmacodynamics, bicalutamide...
    185 KB (20,418 words) - 18:20, 23 September 2024
  • Thumbnail for Ketoconazole
    Ketoconazole (category Nonsteroidal antiandrogens)
    Ketoconazole, sold under the brand name Nizoral among others, is an antiandrogen, antifungal, and antiglucocorticoid medication used to treat a number...
    50 KB (4,379 words) - 21:52, 16 September 2024
  • Thumbnail for Rezvilutamide
    Rezvilutamide (category Nonsteroidal antiandrogens)
    Nonproprietary Name), sold under the brand name Ariane, is a nonsteroidal antiandrogen which is approved for the treatment of prostate cancer in China...
    4 KB (181 words) - 20:06, 30 November 2023
  • Thumbnail for Pyrilutamide
    Pyrilutamide (category Nonsteroidal antiandrogens)
    Pyrilutamide (developmental code name KX-826) is a nonsteroidal antiandrogen (NSAA) – specifically, a selective high-affinity silent antagonist of the...
    8 KB (624 words) - 09:08, 23 September 2024
  • The side effects of bicalutamide, a nonsteroidal antiandrogen (NSAA), including its frequent and rare side effects, have been well-studied and characterized...
    140 KB (15,744 words) - 18:51, 1 September 2024
  • Thumbnail for RU-59063
    N-substituted arylthiohydantoin and was derived from the first-generation nonsteroidal antiandrogen (NSAA) nilutamide. The second-generation NSAAs enzalutamide, RD-162...
    6 KB (496 words) - 21:00, 31 January 2024
  • Darolutamide (category Nonsteroidal antiandrogens)
    asthenia, pain in the arms and legs, and rash. Darolutamide is a nonsteroidal antiandrogen (NSAA), and acts as a selective antagonist of the androgen receptor...
    42 KB (4,162 words) - 00:12, 15 September 2024
  • Thumbnail for AA560
    AA560 (category Nonsteroidal antiandrogens)
    AA560 is an orally active nonsteroidal antiandrogen (NSAA) that was developed in Japan and was first described in the literature in 1977 but was never...
    4 KB (223 words) - 21:02, 15 March 2024
  • Thumbnail for Bicalutamide
    Bicalutamide (category Nonsteroidal antiandrogens)
    recommended during treatment. Bicalutamide is a member of the nonsteroidal antiandrogen (NSAA) group of medications. It works by selectively blocking...
    217 KB (21,643 words) - 16:21, 15 September 2024