• that the others alpha-1 blockers work in a similar manner, since Tamsulosin is an alpha-1-a blocker and Prazosin is an alpha-1 blocker. The risk for floppy...
    38 KB (4,243 words) - 20:56, 27 November 2023
  • Thumbnail for Alpha blocker
    with some β activity. However, the most common type of alpha blocker is usually an α1 blocker. Non-selective α-adrenergic receptor antagonists include:...
    34 KB (3,210 words) - 03:56, 22 March 2024
  • development of beta-3 blocker. Therefore, there is not much information regarding the toxic effect of beta-3 blocker. Alpha-1 blockers such as Alfuzosin,...
    38 KB (3,685 words) - 04:04, 9 June 2024
  • Alpha-2 blockers (or α2 blockers) are a subset of the alpha blocker class of drugs and are antagonists to the α2 adrenergic receptor. They are mainly...
    3 KB (315 words) - 21:37, 9 March 2024
  • Thumbnail for Beta blocker
    β-blocker-induced bronchospasm where it exerts greater efficacy on reversing selective β-blocker-induced bronchospasm than the nonselective β-blocker-induced...
    72 KB (7,108 words) - 07:21, 15 July 2024
  • inhibitors (SSRIs) (e.g., paroxetine, citalopram, sertraline), the alpha-1 blocker silodosin, and anxiolytics. Medications have been associated with spontaneous...
    4 KB (360 words) - 02:54, 18 December 2022
  • clinical uses. Butoxamine, an example of a beta 2 blocker, is only used in research. Alpha 1 blockers prevent smooth muscle contraction by inhibiting the...
    18 KB (1,925 words) - 05:54, 29 November 2023
  • Thumbnail for Tamsulosin
    Tamsulosin (category Alpha-1 blockers)
    Tamsulosin is an alpha blocker and works by relaxing muscles in the prostate. Specifically it is an α1 adrenergic receptor blocker. Tamsulosin was approved...
    17 KB (1,425 words) - 08:26, 1 July 2024
  • Thumbnail for Terazosin
    Terazosin (category Alpha-1 blockers)
    Prostate cancer should be ruled out before starting treatment. It is an alpha-1 blocker and works by relaxing blood vessels and the opening of the bladder...
    5 KB (339 words) - 18:13, 16 April 2024
  • Thumbnail for Alpha-adrenergic agonist
    α2. Alpha 2 receptors are associated with sympatholytic properties. Alpha-adrenergic agonists have the opposite function of alpha blockers. Alpha adrenoreceptor...
    13 KB (1,364 words) - 06:38, 1 April 2024
  • Thumbnail for Carvedilol
    Carvedilol (category Alpha-1 blockers)
    those with liver problems. Carvedilol is a nonselective beta blocker and alpha-1 blocker. How it improves outcomes is not entirely clear but may involve...
    30 KB (2,614 words) - 05:33, 20 May 2024
  • 1098–1104. doi:10.1056/NEJMoa011110. PMID 11596589. "FDA: Manufacturers of TNF-Blocker Drugs Must Highlight Risk of Fungal Infections" (Press release). U.S. Food...
    33 KB (3,686 words) - 07:30, 20 May 2024
  • Thumbnail for Doxazosin
    Doxazosin (redirect from Cardura-1)
    an irregular heart beat, and priapism. It is a α1-selective adrenergic blocker in the quinazoline class of compounds. Doxazosin was patented in 1977 and...
    13 KB (1,006 words) - 13:16, 3 July 2024
  • Thumbnail for Prazosin
    Prazosin (category Alpha-1 blockers)
    nightmares related to post-traumatic stress disorder (PTSD). It is an α1 blocker. It is a less preferred treatment of high blood pressure. Other uses may...
    21 KB (1,778 words) - 14:23, 29 May 2024
  • to which exposure therapy is included in the protocol". Prazosin (alpha-1 blocker) appears useful in decreasing the number of nightmares and the distress...
    23 KB (2,499 words) - 19:36, 21 July 2024
  • Thumbnail for Eugenodilol
    Eugenodilol (category Alpha-1 blockers)
    Eugenodilol is an alpha-1 blocker and beta blocker with weak β2-adrenergic receptor agonist activity derived from eugenol. Huang YC, Wu BN, Lin YT, Chen...
    2 KB (74 words) - 12:38, 13 August 2023
  • Thumbnail for Labetalol
    Labetalol (category Alpha-1 blockers)
    antagonist of the α1-adrenergic receptor, and hence is additionally an alpha blocker. The antagonism of the adrenergic receptors by labetalol is competitive...
    24 KB (2,102 words) - 17:21, 12 May 2024
  • Thumbnail for Amitriptyline
    Amitriptyline (category Alpha-1 blockers)
    Punke MA, Friederich P (May 2007). "Amitriptyline is a potent blocker of human Kv1.1 and Kv7.2/7.3 channels". Anesthesia and Analgesia. 104 (5): 1256–64...
    92 KB (8,667 words) - 10:57, 23 July 2024
  • Thumbnail for Silodosin
    Silodosin (category Alpha-1 blockers)
    the symptomatic treatment of benign prostatic hyperplasia. It acts as an alpha-1 adrenergic receptor antagonist. The most common side effect is a reduction...
    15 KB (1,151 words) - 07:52, 8 May 2024
  • Thumbnail for Naftopidil
    Naftopidil (category Alpha-1 blockers)
    as a selective α1-adrenergic receptor antagonist or alpha-1 blocker. The reaction of 1-naphthol (1) with epichlorohydrin (2) in the presence of alkali...
    4 KB (199 words) - 04:46, 13 July 2024
  • alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are...
    16 KB (1,528 words) - 10:28, 23 June 2024
  • Thumbnail for Dapiprazole
    Dapiprazole (category Alpha-1 blockers)
    Dapiprazole (brand name Rev-Eyes) is an alpha-1 blocker. It is used to reverse mydriasis after eye examination. Doughty MJ, Lyle WM (May 1992). "A review...
    2 KB (65 words) - 04:24, 4 November 2022
  • Thumbnail for Bradycardia
    antihypertensive agent hydralazine, the alpha-1 blocker prazosin, anticholinergics, and sympathomimetic agents like beta-1 agonists. However, side effects, like...
    39 KB (4,428 words) - 00:34, 23 July 2024
  • receptors α-1-Adrenoceptor, an adrenergic receptor with the primary effect of vasoconstriction Alpha-1 blocker, a variety of drugs which block α1-adrenergic...
    5 KB (667 words) - 18:06, 14 March 2022
  • Thumbnail for Phenoxybenzamine
    Phenoxybenzamine (category Alpha-1 blockers)
    names Dibenzyline and Dibenyline) is a non-selective, irreversible alpha blocker. It is used in the treatment of hypertension, and specifically that...
    11 KB (1,021 words) - 20:12, 27 October 2023
  • Thumbnail for Fenspiride
    Fenspiride (category Alpha-1 blockers)
    and torsades de pointes. Fenspiride is known to have activity as an alpha-1 blocker, H1 antagonist, it also inhibits PDE3, PDE4, PDE5 with -logIC50 values...
    4 KB (241 words) - 08:20, 23 February 2024
  • Thumbnail for Quinidine
    Quinidine (category Alpha-1 blockers)
    Quinidine also blocks certain voltage-gated potassium channels (e.g., Kv1.4, Kv4.2, hERG, among others), acts as an antimuscarinic and alpha-1 blocker, and is...
    19 KB (1,862 words) - 01:53, 8 April 2024
  • Thumbnail for Alfuzosin
    Alfuzosin (category Alpha-1 blockers)
    under the brand name Uroxatral among others, is a medication of the α1 blocker class. It is used to treat benign prostatic hyperplasia (BPH). As an antagonist...
    9 KB (710 words) - 08:19, 11 June 2024
  • Thumbnail for Aripiprazole
    Aripiprazole (category Alpha-1 blockers)
    There are studies to date confirming aripiprazole as an antagonist at alpha-adrenergic receptors such as α1A, α2A and α2C, the orthostatic hypotension...
    105 KB (9,711 words) - 08:31, 21 July 2024
  • Thumbnail for Quetiapine
    Quetiapine (category Alpha-1 blockers)
    quetiapine acts primarily as a histamine receptor blocker (antihistamine) and α1-adrenergic blocker. When the dose is increased, quetiapine activates...
    79 KB (6,533 words) - 11:42, 20 June 2024