Selective androgen receptor modulators (SARMs) are a class of drugs that selectively activate the androgen receptor in specific tissues, promoting muscle...
75 KB (6,812 words) - 06:11, 23 October 2024
Antiandrogen (redirect from Androgen receptor antagonist)
for instance androgens and anabolic steroids (AAS) like testosterone, DHT, and nandrolone and selective androgen receptor modulators (SARMs) like enobosarm...
159 KB (15,079 words) - 03:50, 2 November 2024
A selective progesterone receptor modulator (SPRM) is an agent that acts on the progesterone receptor (PR), the biological target of progestogens like...
47 KB (5,150 words) - 12:24, 20 September 2024
Selective glucocorticoid receptor agonists. Selective receptor modulator Selective androgen receptor modulator Selective estrogen receptor modulator Selective...
25 KB (2,554 words) - 14:33, 2 November 2024
of selective estrogen receptor modulators Selective androgen receptor modulator Selective estrogen receptor degrader Selective receptor modulator Timeline...
56 KB (6,362 words) - 22:03, 21 October 2024
Enobosarm (category Selective androgen receptor modulators)
MK-2866, and S-22, is a selective androgen receptor modulator (SARM) which is under development for the treatment of androgen receptor-positive breast cancer...
116 KB (12,937 words) - 22:13, 22 October 2024
The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding...
87 KB (9,390 words) - 08:13, 25 October 2024
allosteric modulators, Examples of receptor modulators in modern medicine include CFTR modulators, selective androgen receptor modulators (SARMs), and...
8 KB (982 words) - 01:08, 20 September 2024
Vosilasarm (category Selective androgen receptor modulators)
and by the black-market name Testolone or Testalone, is a selective androgen receptor modulator (SARM) which is under development for the treatment of hormone-sensitive...
27 KB (2,530 words) - 11:05, 5 March 2024
Classes of selective receptor modulators include: Selective androgen receptor modulator (SARM) Selective estrogen receptor modulator (SERM) Selective glucocorticoid...
2 KB (159 words) - 22:30, 4 October 2023
Ligandrol (category Selective androgen receptor modulators)
name VK5211 and by the black-market name Ligandrol, is a selective androgen receptor modulator (SARM) which is under development for the treatment of muscle...
55 KB (5,985 words) - 21:57, 25 May 2024
YK-11 (category Selective androgen receptor modulators)
synthetic steroidal selective androgen receptor modulator (SARM). It is a gene-selective partial agonist of the androgen receptor (AR) and does not induce...
4 KB (244 words) - 15:55, 28 October 2024
pharmacodynamics, bicalutamide acts as a selective antagonist of the androgen receptor (AR), the biological target of androgens like testosterone and dihydrotestosterone...
186 KB (20,539 words) - 23:49, 10 November 2024
This article pertains to steroidal androgens; nonsteroidal androgens like the selective androgen receptor modulators (SARMs) andarine and enobosarm (ostarine)...
25 KB (654 words) - 12:32, 26 October 2024
Andarine (category Selective androgen receptor modulators)
Andarine (developmental code names GTx-007, S-4) is a selective androgen receptor modulator (SARM) which was developed by GTX, Inc for the treatment of...
10 KB (960 words) - 22:09, 22 October 2024
maintenance of male characteristics in vertebrates by binding to androgen receptors. This includes the embryological development of the primary male sex...
29 KB (3,167 words) - 22:17, 30 October 2024
S-23 (drug) (category Selective androgen receptor modulators)
investigational selective androgen receptor modulator (SARM) developed by GTX, Inc as a potential male hormonal contraceptive. It binds to the androgen receptor more...
3 KB (173 words) - 19:04, 7 January 2023
AC-262,536 (category Selective androgen receptor modulators)
drug developed by Acadia Pharmaceuticals which acts as a selective androgen receptor modulator (SARM). Chemically it possesses endo-exo isomerism, with...
4 KB (308 words) - 21:05, 8 February 2024
Anabolic steroid (redirect from Artificial androgen)
and androgens have been found to increase abdominal fat in postmenopausal women and transgender men as well. Selective androgen receptor modulator Antiandrogen...
209 KB (21,570 words) - 20:09, 4 November 2024
Sex hormone-binding globulin (redirect from Androgen-binding protein)
displace from testosterone 1% or fewer SHBG binding sites. Selective androgen receptor modulators (SARMs) also reduce SHBG. When checking serum estradiol...
57 KB (4,584 words) - 22:43, 2 August 2024
Androgen replacement therapy (ART), often referred to as testosterone replacement therapy (TRT), is a form of hormone therapy in which androgens, often...
25 KB (2,480 words) - 03:42, 2 November 2024
ACP-105 (category Selective androgen receptor modulators)
ACP-105 is a drug which acts as a selective androgen receptor modulator (SARM). It has been investigated for potential use in the treatment of age-related...
4 KB (315 words) - 21:10, 8 February 2024
LGD-3303 (category Selective androgen receptor modulators)
acts as a selective androgen receptor modulator (SARM), with good oral bioavailability. It is a selective agonist for the androgen receptor, producing...
3 KB (203 words) - 20:12, 19 June 2022
to efforts to discover and develop a parallel drug class of selective androgen receptor degraders (SARDs). Fulvestrant requires intramuscular injections...
6 KB (469 words) - 10:25, 3 November 2024
GSK2881078 (category Selective androgen receptor modulators)
GSK2881078 is a drug which acts as a selective androgen receptor modulator (SARM). It was developed for the prevention of muscle wasting and sarcopenia...
3 KB (268 words) - 15:03, 14 January 2024
S-22; VERU-024) – selective androgen receptor modulator for breast cancer [2] GSK-2881078 – selective androgen receptor modulator for cachexia [3] OPK-88004...
15 KB (1,238 words) - 22:37, 30 October 2024
study in rats has shown trenbolone to cause gene expression of the androgen receptor (AR) at least as potent as dihydrotestosterone (DHT). This evidence...
23 KB (1,906 words) - 08:25, 12 July 2024
Nonsteroidal antiandrogen (redirect from Nonsteroidal androgen receptor antagonist)
are typically selective and full or silent antagonists of the androgen receptor (AR) and act by directly blocking the effects of androgens like testosterone...
17 KB (1,576 words) - 15:57, 24 February 2024
MK-0773 (category Selective androgen receptor modulators)
also known as PF-05314882, is a steroidal, orally active selective androgen receptor modulator (SARM) that was under development by Merck and GTx for the...
11 KB (965 words) - 15:54, 28 October 2024
Marieta (February 2023). "Exploring the polymorphism of selective androgen receptor modulator YK11". Journal of Molecular Structure. 1273: 134281....
11 KB (1,195 words) - 00:18, 21 June 2024