that the others alpha-1 blockers work in a similar manner, since Tamsulosin is an alpha-1-a blocker and Prazosin is an alpha-1 blocker. The risk for floppy...
38 KB (4,275 words) - 20:35, 6 October 2024
with some β activity. However, the most common type of alpha blocker is usually an α1 blocker. Non-selective α-adrenergic receptor antagonists include:...
35 KB (3,197 words) - 06:35, 26 October 2024
development of beta-3 blocker. Therefore, there is not much information regarding the toxic effect of beta-3 blocker. Alpha-1 blockers such as Alfuzosin,...
38 KB (3,668 words) - 08:21, 29 October 2024
Alpha-2 blockers (or α2 blockers) are a subset of the alpha blocker class of drugs and are antagonists to the α2 adrenergic receptor. They are mainly...
3 KB (339 words) - 18:58, 20 August 2024
clinical uses. Butoxamine, an example of a beta 2 blocker, is only used in research. Alpha 1 blockers prevent smooth muscle contraction by inhibiting the...
18 KB (1,925 words) - 05:54, 29 November 2023
β-blocker-induced bronchospasm where it exerts greater efficacy on reversing selective β-blocker-induced bronchospasm than the nonselective β-blocker-induced...
75 KB (7,463 words) - 11:05, 14 October 2024
inhibitors (SSRIs) (e.g., paroxetine, citalopram, sertraline), the alpha-1 blocker silodosin, and anxiolytics. Medications have been associated with spontaneous...
4 KB (360 words) - 02:54, 18 December 2022
Tamsulosin (category Alpha-1 blockers)
Tamsulosin is an alpha blocker and works by relaxing muscles in the prostate. Specifically it is an α1-adrenergic receptor blocker. Tamsulosin was approved...
17 KB (1,433 words) - 20:25, 6 October 2024
Terazosin (category Alpha-1 blockers)
Prostate cancer should be ruled out before starting treatment. It is an alpha-1 blocker and works by relaxing blood vessels and the opening of the bladder...
6 KB (340 words) - 20:10, 6 October 2024
Carvedilol (category Alpha-1 blockers)
those with liver problems. Carvedilol is a nonselective beta blocker and alpha-1 blocker. How it improves outcomes is not entirely clear but may involve...
33 KB (2,908 words) - 03:30, 7 September 2024
TNF inhibitor (redirect from TNF alpha blocker)
1098–1104. doi:10.1056/NEJMoa011110. PMID 11596589. "FDA: Manufacturers of TNF-Blocker Drugs Must Highlight Risk of Fungal Infections" (Press release). U.S. Food...
33 KB (3,686 words) - 07:30, 20 May 2024
α2. Alpha 2 receptors are associated with sympatholytic properties. Alpha-adrenergic agonists have the opposite function of alpha blockers. Alpha adrenoreceptor...
13 KB (1,360 words) - 22:27, 10 September 2024
Amitriptyline (category Alpha-1 blockers)
Punke MA, Friederich P (May 2007). "Amitriptyline is a potent blocker of human Kv1.1 and Kv7.2/7.3 channels". Anesthesia and Analgesia. 104 (5): 1256–64...
92 KB (8,729 words) - 03:44, 26 October 2024
Labetalol (category Alpha-1 blockers)
antagonist of the α1-adrenergic receptor, and hence is additionally an alpha blocker. The antagonism of the adrenergic receptors by labetalol is competitive...
29 KB (2,553 words) - 19:03, 2 August 2024
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are...
16 KB (1,528 words) - 10:28, 23 June 2024
Prazosin (category Alpha-1 blockers)
nightmares related to post-traumatic stress disorder (PTSD). It is an α1 blocker. It is a less preferred treatment of high blood pressure. Other uses may...
21 KB (1,776 words) - 04:42, 9 October 2024
to which exposure therapy is included in the protocol". Prazosin (alpha-1 blocker) appears useful in decreasing the number of nightmares and the distress...
23 KB (2,499 words) - 21:12, 25 October 2024
Trimazosin (category Alpha-1 blockers)
Trimazosin is a sympatholytic alpha-1 blocker. van Kalken CK, van der Meulen J, Oe PL, Vriesendorp R, Donker AJ (1986). "Pharmacokinetics of trimazosin...
3 KB (69 words) - 15:06, 1 September 2022
Silodosin (category Alpha-1 blockers)
the symptomatic treatment of benign prostatic hyperplasia. It acts as an alpha-1 adrenergic receptor antagonist. The most common side effect is a reduction...
15 KB (1,151 words) - 20:15, 6 October 2024
Clozapine (category Alpha-1 blockers)
Clozapine?". Clinical Schizophrenia & Related Psychoses. 1 (1): 92–95. doi:10.3371/csrp.1.1.8. Downs J, Zinkler M (October 2007). "Clozapine: national...
136 KB (14,536 words) - 03:47, 26 October 2024
Phenoxybenzamine (category Alpha-1 blockers)
names Dibenzyline and Dibenyline) is a non-selective, irreversible alpha blocker. It is used in the treatment of hypertension, and specifically that...
11 KB (1,021 words) - 20:12, 27 October 2023
Trazodone (category Alpha-1 blockers)
human targets in question. Roughly half of brain 5-HT2A receptors are blocked by 1 mg of trazodone and essentially all 5-HT2A receptors are saturated at...
115 KB (10,960 words) - 16:04, 2 November 2024
Dapiprazole (category Alpha-1 blockers)
Dapiprazole (brand name Rev-Eyes) is an alpha-1 blocker. It is used to reverse mydriasis after eye examination. Doughty MJ, Lyle WM (May 1992). "A review...
2 KB (65 words) - 20:12, 30 August 2024
Quetiapine (category Alpha-1 blockers)
quetiapine acts primarily as a histamine receptor blocker (antihistamine) and α1-adrenergic blocker. When the dose is increased, quetiapine activates...
79 KB (6,427 words) - 19:30, 7 October 2024
Alfuzosin (category Alpha-1 blockers)
under the brand name Uroxatral among others, is a medication of the α1 blocker class. It is used to treat benign prostatic hyperplasia (BPH). As an antagonist...
9 KB (710 words) - 20:17, 6 October 2024
Olanzapine (category Alpha-1 blockers)
serotonin2, muscarinic, histamine H1 and alpha 1-adrenergic receptors in vitro". Schizophrenia Research. 37 (1): 107–122. doi:10.1016/s0920-9964(98)00146-7...
97 KB (9,053 words) - 06:06, 31 October 2024
List of A1 genes, proteins or receptors (redirect from Alpha 1 gene)
receptors α-1-Adrenoceptor, an adrenergic receptor with the primary effect of vasoconstriction Alpha-1 blocker, a variety of drugs which block α1-adrenergic...
5 KB (667 words) - 18:06, 14 March 2022
Aripiprazole (category Alpha-1 blockers)
There are studies to date confirming aripiprazole as an antagonist at alpha-adrenergic receptors such as α1A, α2A and α2C, the orthostatic hypotension...
106 KB (9,750 words) - 20:06, 22 October 2024
Quinidine (category Alpha-1 blockers)
Quinidine also blocks certain voltage-gated potassium channels (e.g., Kv1.4, Kv4.2, hERG, among others), acts as an antimuscarinic and alpha-1 blocker, and is...
19 KB (1,911 words) - 11:25, 5 November 2024