A serotonin receptor agonist is an agonist of one or more serotonin receptors. They activate serotonin receptors in a manner similar to that of serotonin...
16 KB (1,662 words) - 21:10, 6 November 2024
5-HT receptors, 5-hydroxytryptamine receptors, or serotonin receptors, are a group of G protein-coupled receptor and ligand-gated ion channels found in...
65 KB (5,263 words) - 07:14, 24 November 2024
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). The 5-HT2A...
91 KB (9,998 words) - 02:42, 25 November 2024
A serotonin antagonist, or serotonin receptor antagonist, is a drug used to inhibit the action of serotonin and serotonergic drugs at serotonin (5-HT)...
5 KB (503 words) - 03:53, 9 October 2024
which acts as a serotonin reuptake inhibitor (SRI), agonist of the 5-HT1A receptor, and antagonist of the 5-HT3 and 5-HT7 receptors. However, it can...
5 KB (568 words) - 17:03, 21 March 2024
tandospirone act as serotonin 5-HT1A receptor agonists. Many antipsychotics bind to and modulate serotonin receptors, including the serotonin 5-HT1A, 5-HT2A...
156 KB (16,610 words) - 13:36, 19 November 2024
The serotonin 1A receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter...
58 KB (6,188 words) - 15:33, 22 September 2024
Lisuride (category Serotonin receptor agonists)
Lisuride acts as a mixed agonist and antagonist of dopamine, serotonin, and adrenergic receptors. Activation of specific dopamine receptors is thought to be responsible...
27 KB (2,110 words) - 00:27, 26 October 2024
5-hydroxytryptamine (serotonin) receptor 1D, also known as HTR1D, is a 5-HT receptor, but also denotes the human gene encoding it. 5-HT1D acts on the...
11 KB (1,238 words) - 09:14, 27 October 2024
(serotonin) receptor 5A, also known as HTR5A, is a protein that in humans is encoded by the HTR5A gene. Agonists and antagonists for 5-HT receptors, as...
15 KB (1,674 words) - 17:31, 10 November 2024
non-competitive NMDA receptor antagonist α-Methyltryptamine [αMT] (Indopan) – non-selective serotonin receptor agonist, serotonin–norepinephrine–dopamine...
18 KB (1,531 words) - 05:27, 18 November 2024
5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT2B is a member...
50 KB (5,105 words) - 09:12, 25 November 2024
A GABA receptor agonist is a drug that is an agonist for one or more of the GABA receptors, producing typically sedative effects, and may also cause other...
8 KB (749 words) - 21:06, 6 November 2024
LY-2456302) – κ-opioid receptor antagonist CYB003 (CYB-003; deuterated psilocybin analogue) – serotonin 5-HT2A receptor agonist and psychedelic hallucinogen...
146 KB (11,183 words) - 01:32, 25 November 2024
Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has two subclasses...
13 KB (1,359 words) - 20:52, 24 November 2024
5-MeO-DMT (category Serotonin receptor agonists)
The drug acts as a non-selective serotonin receptor agonist, including of the serotonin 5-HT1A and 5-HT2A receptors among others. However, 5-MeO-DMT differs...
36 KB (3,173 words) - 21:45, 13 November 2024
this class as it does not function as a serotonin antagonist, acting solely as a 5-HT1A receptor partial agonist instead. Vortioxetine (Trintellix) – another...
9 KB (615 words) - 21:41, 9 March 2024
agonists of the beta receptors are selective for one or more beta-adrenoreceptors. For example, patients with low heart rate are given beta agonist treatments...
10 KB (851 words) - 21:05, 24 November 2024
activates that receptor. For example, the endogenous agonist for serotonin receptors is serotonin, and the endogenous agonist for dopamine receptors is dopamine...
14 KB (1,622 words) - 03:21, 4 September 2024
Later, animal studies showed that serotonin receptor agonists might act as a mediator of satiety. Serotonin has been implicated as a critical factor in...
48 KB (5,032 words) - 18:40, 8 March 2024
Beta2-adrenergic agonists, also known as adrenergic β2 receptor agonists, are a class of drugs that act on the β2 adrenergic receptor. Like other β adrenergic...
18 KB (1,703 words) - 06:18, 17 March 2024
A muscarinic acetylcholine receptor agonist, also simply known as a muscarinic agonist or as a muscarinic agent, is an agent that activates the activity...
9 KB (858 words) - 23:25, 21 November 2024
Tryptamine (category Serotonin receptor agonists)
specific to tryptamine degradation. Tryptamine is known to act as a serotonin receptor agonist, although its potency is limited by rapid inactivation by monoamine...
54 KB (4,458 words) - 05:16, 25 November 2024
5-MeO-MiPT (category Serotonin receptor agonists)
effects. The drug acts as a non-selective serotonin receptor agonist, including of the serotonin 5-HT2A receptor. 5-MeO-MiPT is in a class of compounds commonly...
18 KB (1,383 words) - 03:10, 22 November 2024
N-Methyltryptamine (category Serotonin receptor agonists)
5-methoxy-N,N-dimethyltryptamine (5-MeO-DMT). NMT acts as a serotonin receptor agonist and serotonin releasing agent and produces psychoactive and hallucinogenic...
8 KB (643 words) - 09:14, 2 November 2024
receptor rather than activating it like an agonist. Antagonist drugs interfere in the natural operation of receptor proteins. They are sometimes called blockers;...
33 KB (3,845 words) - 01:47, 19 August 2024
A dopamine agonist is a compound that activates dopamine receptors. There are two families of dopamine receptors, D1-like and D2-like. They are all G...
44 KB (5,009 words) - 23:25, 21 November 2024
(MDMA; "ecstasy") – serotonin, norepinephrine, and dopamine releasing agent, weak serotonin 5-HT2A, 5-HT2B, 5-HT2C receptor agonist, entactogen, and weak...
92 KB (7,758 words) - 02:13, 18 November 2024
"Entrez Gene: HTR1B 5-hydroxytryptamine (serotonin) receptor 1B". "5-hydroxytryptamine (serotonin) receptor 1B, G protein-coupled". Retrieved 23 Feb 2013...
17 KB (1,984 words) - 08:01, 27 October 2024
The 5HT6 receptor is a subtype of 5HT receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5HT). It is a G protein-coupled...
29 KB (3,308 words) - 15:33, 22 September 2024