Tipifarnib (INN,: 213 proposed trade name Zarnestra) is a farnesyltransferase inhibitor. Farnesyltransferase inhibitors block the activity of the farnesyltransferase...
9 KB (673 words) - 08:55, 9 September 2024
(Lonafarnib) was the first to do so, followed by R115777 (Zarnestra, Tipifarnib). Unfortunately, the predicted "early potential [of FTIs] has not been...
12 KB (1,079 words) - 17:42, 26 May 2021
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
11 KB (734 words) - 02:39, 12 October 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
31 KB (2,908 words) - 06:38, 22 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
36 KB (3,278 words) - 07:36, 30 September 2024
toothpaste Rolaids RWJ-51204 Savlon Sinutab Splenda Sylvant Telaprevir Tipifarnib Buildings Johnson and Johnson Plaza Related 2010 DePuy Hip Recall 2010...
7 KB (764 words) - 16:32, 18 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
15 KB (1,438 words) - 02:57, 10 May 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
61 KB (6,086 words) - 21:24, 28 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
4 KB (411 words) - 21:05, 6 May 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
79 KB (9,506 words) - 01:11, 14 July 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
14 KB (1,105 words) - 06:03, 14 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
19 KB (1,681 words) - 07:11, 15 March 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
18 KB (1,467 words) - 23:44, 20 August 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
20 KB (1,809 words) - 14:07, 16 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
9 KB (716 words) - 09:40, 4 August 2024
Crucell was renamed as Janssen Vaccines. In March 2015, Janssen licensed tipifarnib (a farnesyl transferase inhibitor) to Kura Oncology who will assume sole...
33 KB (3,169 words) - 05:41, 1 October 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
60 KB (6,445 words) - 15:35, 26 September 2024
inhibits fibroblast growth. Studies showed no improvement over controls. Tipifarnib (also known as drug R115777) inhibits the activation of RAS. This drug...
30 KB (3,257 words) - 22:04, 21 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
16 KB (1,041 words) - 22:27, 20 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
52 KB (708 words) - 12:37, 26 August 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
9 KB (595 words) - 06:22, 6 October 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
26 KB (2,647 words) - 18:18, 22 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
14 KB (1,009 words) - 23:04, 20 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
49 KB (4,454 words) - 18:07, 8 August 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
16 KB (1,230 words) - 04:49, 15 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
24 KB (2,132 words) - 11:10, 7 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
39 KB (3,990 words) - 01:39, 28 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
39 KB (3,864 words) - 22:43, 20 September 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
13 KB (1,449 words) - 12:45, 21 August 2024
Enzyme inhibitors FI (Tipifarnib§) CDK inhibitors (Abemaciclib Alvocidib† Palbociclib Ribociclib Seliciclib†) PrI Bortezomib Carfilzomib Oprozomib Ixazomib...
6 KB (302 words) - 01:44, 27 August 2024