Estrogen receptor beta (ERβ) also known as NR3A2 (nuclear receptor subfamily 3, group A, member 2) is one of two main types of estrogen receptor—a nuclear...
39 KB (4,526 words) - 06:00, 25 July 2024
Estrogen receptors (ERs) are proteins found in cells that function as receptors for the hormone estrogen (17β-estradiol). There are two main classes of...
38 KB (4,058 words) - 04:20, 19 October 2024
Estrogen receptor alpha (ERα), also known as NR3A1 (nuclear receptor subfamily 3, group A, member 1), is one of two main types of estrogen receptor, a...
58 KB (6,133 words) - 06:55, 2 November 2024
Estrogen-related receptor beta (ERR-β), also known as ESRRB or NR3B2 (nuclear receptor subfamily 3, group B, member 2), is a nuclear receptor that in...
7 KB (800 words) - 19:11, 27 March 2024
Selective estrogen receptor modulators (SERMs), also known as estrogen receptor agonists/antagonists (ERAAs), are a class of drugs that act on estrogen receptors...
56 KB (6,362 words) - 22:03, 21 October 2024
Erteberel (redirect from Selective estrogen receptor beta agonist-1)
LY-500307; also known as selective estrogen receptor beta agonist-1 or SERBA-1) is a synthetic, nonsteroidal estrogen which acts as a selective ERβ agonist...
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mediated by binding to two receptors: Estrogen Receptor alpha (ERα) and Estrogen Receptor beta (ERβ). These two receptors are tissue specific and have...
19 KB (2,223 words) - 00:10, 29 October 2024
physical performance. In humans, it is hypothesized to bind to the estrogen receptor beta (ERβ) protein-coding gene. The primary sources of 20-hydroxyecdysone...
13 KB (1,152 words) - 10:34, 24 September 2024
SERBA-2 (redirect from Selective estrogen receptor beta agonist-2)
SERBA-2, short for selective estrogen receptor beta agonist-2, is a synthetic, nonsteroidal estrogen which acts as a selective ERβ agonist. For the ERα...
4 KB (291 words) - 06:49, 21 August 2022
Estradiol (redirect from 17-beta estradiol)
PMID 21839626. Thomas CG, Strom A, Lindberg K, Gustafsson JA (June 2011). "Estrogen receptor beta decreases survival of p53-defective cancer cells after DNA damage...
75 KB (7,243 words) - 18:59, 30 October 2024
Equol (section Estrogen receptor binding)
binding affinity for human estrogen receptor alpha (ERα) and 20% of estradiol's binding affinity for human estrogen receptor beta (ERβ). The preferential...
24 KB (2,667 words) - 21:44, 28 February 2024
estrogen receptor (ER): estrogen receptor alpha (ERα), and estrogen receptor beta (ER-β), also known as NR3A2. Both are nuclear receptors activated by the sex...
10 KB (1,332 words) - 19:38, 30 June 2024
tremors. Beta adrenergic receptor kinase Beta adrenergic receptor kinase-2 Acetylcholine receptor (Cholinergic receptor) Nicotinic acetylcholine receptor Muscarinic...
33 KB (2,982 words) - 11:42, 7 August 2024
selective estrogen receptor beta agonist for hot flashes associated with menopause Seala (formerly VG101) a selective estrogen receptor beta agonist for...
10 KB (987 words) - 15:39, 14 November 2022
with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones. There are three human estrogen related receptors: ERRα...
11 KB (1,175 words) - 13:05, 3 December 2023
studied steroid hormone receptors are members of the nuclear receptor subfamily 3 (NR3) that include receptors for estrogen (group NR3A) and 3-ketosteroids...
23 KB (2,796 words) - 19:08, 19 February 2024
The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...
33 KB (3,418 words) - 06:46, 20 October 2024
nuclear receptors include members of subfamily 3, such as the androgen receptor, estrogen receptors, glucocorticoid receptor, and progesterone receptor. It...
74 KB (6,683 words) - 09:55, 12 September 2024
they bind to and activate estrogen receptors (ERs) which in turn modulate the expression of many genes. Additionally, estrogens bind to and activate rapid-signaling...
73 KB (7,787 words) - 14:58, 29 October 2024
Hong SS, Hwang DJ, Miller DD, Dalton JT (2010). "Estrogen receptor beta selective nonsteroidal estrogens: seeking clinical indications". Expert Opin Ther...
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PMID 25938107. Isgor C, Cecchi M, Kabbaj M, Akil H, Watson SJ (2003). "Estrogen receptor beta in the paraventricular nucleus of hypothalamus regulates the neuroendocrine...
50 KB (4,977 words) - 18:21, 31 August 2024
Estrogen-related receptor alpha (ERRα), also known as NR3B1 (nuclear receptor subfamily 3, group B, member 1), is a nuclear receptor that in humans is...
17 KB (1,995 words) - 21:24, 29 March 2024
The beta-1 adrenergic receptor (β1 adrenoceptor), also known as ADRB1, can refer to either the protein-encoding gene (gene ADRB1) or one of the four adrenergic...
31 KB (3,742 words) - 16:12, 25 October 2024
identified, including NQO2 (alone and in interaction with AKT1), GSTP1, estrogen receptor beta, CBR1, and integrin αVβ. It was unclear at that time if any or all...
41 KB (3,914 words) - 10:47, 25 September 2024
Erb's muscular dystrophy, or simply Erb's Estrogen receptor beta (ERβ), one of two main types of estrogen receptors Effective resolution bandwidth Equivalent...
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Androgen receptors Calcitriol receptors Corticotropin-releasing hormone receptor 1 Corticotropin releasing hormone receptor 2 Estrogen receptors Follicle-stimulating...
17 KB (2,005 words) - 23:01, 20 August 2024
3β-Androstanediol (category Estrogens)
Edinger, K; Osborne, D; Walf, A (2008). "Androgens with activity at estrogen receptor beta have anxiolytic and cognitive-enhancing effects in male rats and...
13 KB (1,266 words) - 22:20, 3 December 2023
Luteinizing hormone (redirect from Receptors, lh)
growth, specifically affecting granulosa cells. With the rise in estrogens, LH receptors are also expressed on the maturing follicle, which causes it to...
34 KB (3,380 words) - 21:31, 24 October 2024
Albert LM, Leathurby Y, et al. (October 2003). "Evaluation of an estrogen receptor-beta agonist in animal models of human disease". Endocrinology. 144 (10):...
4 KB (243 words) - 09:38, 23 April 2022
The beta-3 adrenergic receptor (β3-adrenoceptor), also known as ADRB3, is a beta-adrenergic receptor, and also denotes the human gene encoding it. Actions...
17 KB (2,039 words) - 09:45, 7 October 2023