Gabapentin, sold under the brand name Neurontin among others, is an anticonvulsant medication primarily used to treat partial seizures and neuropathic...
91 KB (8,944 words) - 03:28, 14 August 2024
gabapentin. It was designed for increased oral bioavailability over gabapentin, and human trials showed it to produce extended release of gabapentin with...
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United States in 2004. It was developed as a successor to the related gabapentin. It is available as a generic medication. In 2021, it was the 73rd most...
99 KB (8,544 words) - 08:10, 2 August 2024
the gabapentin receptor (α2δ subunit), as it is the target of the drugs gabapentin and pregabalin. Clinically used gabapentinoids include gabapentin, pregabalin...
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seizures and severe agitation. Approved: Gabapentin (Neurontin) Gabapentin enacarbil (Horizant, Regnite) Gabapentin Extended-Release (Gralise) Pregabalin...
130 KB (13,449 words) - 03:44, 19 August 2024
disorder. Curry, W. J; Kulling, D. L (1998). "Newer antiepileptic drugs: Gabapentin, lamotrigine, felbamate, topiramate and fosphenytoin". American Family...
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used transdermally (applied topically to the skin) in combination with gabapentin and clonidine prepared at a compounding pharmacy. Common side effects...
34 KB (3,272 words) - 19:55, 10 August 2024
most widely attempted medication is gabapentin, with one case series finding that seven of eight patients on gabapentin showed improvement in attack frequency...
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Phenibut also binds to and blocks α2δ subunit-containing VDCCs, similarly to gabapentin and pregabalin, and hence is a gabapentinoid. Both (R)-phenibut and (S)-phenibut...
36 KB (2,858 words) - 14:31, 24 August 2024
4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...
177 KB (18,939 words) - 12:01, 23 August 2024
4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...
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to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was developed as a potentially more potent successor to gabapentin and...
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Pregabalin (2004) Mirogabalin (2019) (Japan only) Gabapentin (1993) Gabapentin enacarbil (Horizant) (2011) Gabapentin extended release (Gralise) (1996) Gabapentinoids...
70 KB (5,714 words) - 02:50, 19 August 2024
dopamine agonists like pramipexole and gabapentinoids (α2δ ligands) like gabapentin. RLS affects an estimated 2.5–15% of the American population. Females...
79 KB (8,316 words) - 13:15, 16 August 2024
anti-convulsant medications gabapentin and pregabalin may be used to reduce pain. There is tentative evidence that gabapentin may be of benefit for pain...
168 KB (17,868 words) - 16:04, 23 August 2024
short trial period of gabapentin therapy is recommended, to determine the effectiveness for that person. 62% of people taking gabapentin may have at least...
59 KB (6,666 words) - 12:55, 24 August 2024
hot flashes include cognitive-behavioral therapy, clinical hypnosis, gabapentin, fezolinetant or selective serotonin reuptake inhibitors. These will not...
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severe allergic reactions due to its strong antihistamine properties. Gabapentin, approved for treatment of seizures and postherpetic neuralgia in adults...
13 KB (1,254 words) - 23:52, 6 July 2024
fingers in lidocaine; milk or vinegar; or the use of local nerve blocks, gabapentin, or topical corticosteroids. Hunan hand can be prevented by wearing rubber...
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advantage over certain anxiolytic medications such as benzodiazepines. Gabapentin (Neurontin), a closely related medication to pregabalin with the same...
111 KB (14,516 words) - 19:33, 24 August 2024
inhibitor and GABA reuptake inhibitor Gabapentin – anticonvulsant; inhibitor of α2δ subunit-containing VGCCs Gabapentin enacarbil – used for the treatment...
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dissociative anesthetic used in surgery) is useful in bipolar disorder. Gabapentin and pregabalin are not proven to be effective for treating bipolar disorder...
156 KB (17,555 words) - 17:03, 17 August 2024
non-steroidal anti-inflammatory drugs (NSAIDs), prostaglandin-based drugs, gabapentin, and methylcobalamin. However, the quality of evidence supporting their...
60 KB (6,696 words) - 11:35, 23 August 2024
Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin Antidepressants SSRIsTooltip Selective...
87 KB (7,810 words) - 06:35, 18 August 2024
pharmaceutical marketing. In 1993, the Food and Drug Administration (FDA) approved gabapentin only for treatment of seizures. Warner–Lambert, which merged with Pfizer...
168 KB (14,563 words) - 23:11, 15 August 2024
Development Ltd. acquired the exclusive rights to develop and commercialize Gabapentin ER. The drug had been developed by DDL. 2003 saw a net loss of $30 million...
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with newer anti-seizure medications such as gabapentin, offer a possible regimen for seizure control. Gabapentin has the additional feature of aiding in the...
64 KB (6,616 words) - 12:51, 17 August 2024
bowel or bladder function. Many treatments, including corticosteroids, gabapentin, pregabalin, acupuncture, heat or ice, and spinal manipulation, have limited...
46 KB (5,037 words) - 20:26, 11 August 2024
Calcium blockers Alcohol (ethanol) Gabapentin Gabapentin enacarbil Leconotide Mirogabalin Pregabalin Ziconotide Sodium blockers Carbamazepine Lacosamide...
96 KB (10,049 words) - 16:46, 23 August 2024
consisting of a combination of hydroxyzine and two other medications (gabapentin and flumazenil) as well as therapy, is an ineffective treatment promoted...
43 KB (3,708 words) - 11:54, 8 July 2024