Phenyltropanes (PTs) are a family of chemical compounds originally derived from structural modification of cocaine. The main feature differentiating phenyltropanes...

List of aminorex analogues List of benzodiazepines List of fentanyl analogues List of phenyltropanes Utopioid Pergolizzi Jr J, Raffa R, LeQuang JA, Breve...

displacement of [3H]paroxetine (5-HTT & NET) bFor displacement of [3H]nisoxetine (5-HTT & NET) See: List of phenyltropanes (Many phenyltropanes are derived...

to the wording on the entry of coca in Schedule 1 of the Controlled Drugs and Substances Act. List of phenyltropanes List of cocaine analogues Amfonelic...

Arylcyclohexylamine List of benzimidazole opioids List of phenyltropanes Structural scheduling of synthetic cannabinoids Substituted cathinone Utopioid Hassanien...

phenyltropanes which were tested in clinical trials. Tesofensine Brasofensine NS-2359 (GSK-372,475) 3,4-DCMP O-2390 List of cocaine analogues List of...

oxatropane tropoxane. List of phenyltropanes Pham-Huu DP, Deschamps JR, Liu S, Madras BK, Meltzer PC (January 2007). "Synthesis of 8-thiabicyclo[3.2.1]octanes...

methylenedioxyphenethylamine List of aminorex analogues List of methylphenidate analogues List of phenyltropanes List of cocaine analogues Boswell GE...

supranuclear palsy. RTI-55 is made as follows: RTI-121 RTI-229 RTI-352 List of Phenyltropanes Boja JW, Patel A, Carroll FI, Rahman MA, Philip A, Lewin AH, et al...

controlled substance analogue of cocaine on the grounds of its related chemical structure. RTI-55 RTI-160 List of Phenyltropanes Carroll FI, Kotian P, Dehghani...

dose. WIN 35,065-2 List of phenyltropanes List of cocaine analogues Wee S, Carroll FI, Woolverton WL (February 2006). "A reduced rate of in vivo dopamine...

demethylation step. See for example the list of phenyltropanes or the synthesis of paroxetine for further examples of this. Diacetylnalorphine Levallorphan...

pronounced effects in terms of speed of onset and rate of stimulation among many differing phenyltropanes. List of phenyltropanes RTI-126 O-4210 Kimmel HL...

substance analogue of cocaine on the grounds of its related chemical structure. RTI-55 List of cocaine analogues List of Phenyltropanes Scheffel U, Dannals...

cocaine compared to longer acting analogues like RTI-121 and RTI-177. List of phenyltropanes RTI-113 Silverthorn ML, Dersch CM, Baumann MH, Cadet JL, Partilla...

Carroll FI, Kuhar MJ (December 2001). "Locomotor stimulant effects of novel phenyltropanes in the mouse". Drug and Alcohol Dependence. 65 (1): 25–36. doi:10...

scaffold to correctly orientate the binding groups, and for each of the hundreds of phenyltropanes that are known, there may be a phenidate equivalent with a...

be caused by lack of BBB penetration, or interactions at alternative receptor sites. List of cocaine analogues List of phenyltropanes Navarro HA, Howard...

is a phenyltropane homologue of paroxetine developed by the group led by F Ivy Carroll in the 1990s. Very few esters of phenyltropanes are actually...

its own derived phenyltropanes analogues which have that removed. In addition to this, cocaine has some target binding to the site of the κ-opioid receptor...

(mostly restricted to various phenyltropanes) RU – Roussel Uclaf RWJ – R.W. Johnson Pharmaceutical Research, now part of Johnson & Johnson SAGE – Sage...

pair of racemers. With a racemic pair of diastereomers, there is still the question of syn (cis) or anti (trans). In the case of the phenyltropanes, although...

among the faster onsets of action from among phenyltropanes) These characteristics make it a potential candidate for treatment of cocaine addiction, as...

substituted phenyltropanes are highly potent MAT inhibitors and also have a very long half-life, spanning perhaps at least a few days; as the half-life of the...

pharmacophore model for cocaine and phenyltropanes comprises two electrostatic interactions of the basic nitrogen and the ester group of the C-2 substituent, and...

that breastfeeding be interrupted for three days after administration. List of cocaine analogues "Neurological therapies". Health Canada. 9 May 2018....

Carroll FI, Kuhar MJ (December 2001). "Locomotor stimulant effects of novel phenyltropanes in the mouse". Drug and Alcohol Dependence. 65 (1): 25–36. doi:10...

monoamine transporter affinity of new 2beta-carbomethoxy-3beta-[4-(substituted thiophenyl)]phenyltropanes: discovery of a selective SERT antagonist with...

cannabinoid EAM-2201 was banned from 6 December 2012. Another stimulant, the phenyltropane derivative RTI-126, was banned from 27 December 2012. Two more cannabinoids...

legislation. List of cocaine analogues Kimmel HL, Carroll FI, Kuhar MJ (December 2001). "Locomotor stimulant effects of novel phenyltropanes in the mouse"...