Gabapentin, sold under the brand name Neurontin among others, is an anticonvulsant medication primarily used to treat partial seizures and neuropathic...

gabapentin. It was designed for increased oral bioavailability over gabapentin, and human trials showed it to produce extended release of gabapentin with...

United States in 2004. It was developed as a successor to the related gabapentin. It is available as a generic medication. In 2022, it was the 91st most...

the gabapentin receptor (α2δ subunit), as it is the target of the drugs gabapentin and pregabalin. Clinically used gabapentinoids include gabapentin, pregabalin...

seizures and severe agitation. Approved: Gabapentin (Neurontin) Gabapentin enacarbil (Horizant, Regnite) Gabapentin Extended-Release (Gralise) Pregabalin...

used transdermally (applied topically to the skin) in combination with gabapentin and clonidine prepared at a compounding pharmacy. Common side effects...

Phenibut also binds to and blocks α2δ subunit-containing VDCCs, similarly to gabapentin and pregabalin, and hence is a gabapentinoid. Both (R)-phenibut and (S)-phenibut...

Pregabalin (2004) Mirogabalin (2019) (Japan only) Gabapentin (1993) Gabapentin enacarbil (Horizant) (2011) Gabapentin extended release (Gralise) (1996) Gabapentinoids...

4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...

inhibitor and GABA reuptake inhibitor Gabapentin – anticonvulsant; inhibitor of α2δ subunit-containing VGCCs Gabapentin enacarbil – used for the treatment...

most widely attempted medication is gabapentin, with one case series finding that seven of eight patients on gabapentin showed improvement in attack frequency...

to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was developed as a potentially more potent successor to gabapentin and...

short trial period of gabapentin therapy is recommended, to determine the effectiveness for that person. 62% of people taking gabapentin may have at least...

4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...

hot flashes include cognitive-behavioral therapy, clinical hypnosis, gabapentin, fezolinetant or selective serotonin reuptake inhibitors. These will not...

advantage over certain anxiolytic medications such as benzodiazepines. Gabapentin (Neurontin), a closely related medication to pregabalin with the same...

anti-convulsant medications gabapentin and pregabalin may be used to reduce pain. There is tentative evidence that gabapentin may be of benefit for pain...

(duloxetine, venlafaxine, and milnacipran) and antiepileptic medications (gabapentin, pregabalin, oxcarbazepine zonisamide levetiracetam, lamotrigine, topiramate...

propanamide does not change after Hofmann reaction. In the synthesis of gabapentin, beginning with the mono-amidation of 1,1-cyclohexane diacetic acid anhydride...

non-steroidal anti-inflammatory drugs (NSAIDs), prostaglandin-based drugs, gabapentin, and methylcobalamin. However, the quality of evidence supporting their...

dopamine agonists like pramipexole and gabapentinoids (α2δ ligands) like gabapentin. RLS affects an estimated 2.5–15% of the American population. Females...

pharmaceutical marketing. In 1993, the Food and Drug Administration (FDA) approved gabapentin only for treatment of seizures. Warner–Lambert, which merged with Pfizer...

Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin Antidepressants SSRIsTooltip Selective...

with newer anti-seizure medications such as gabapentin, offer a possible regimen for seizure control. Gabapentin has the additional feature of aiding in the...

Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin Antidepressants SSRIsTooltip Selective...

Development Ltd. acquired the exclusive rights to develop and commercialize Gabapentin ER. The drug had been developed by DDL. 2003 saw a net loss of $30 million...

Calcium blockers Alcohol (ethanol) Gabapentin Gabapentin enacarbil Leconotide Mirogabalin Pregabalin Ziconotide Sodium blockers Carbamazepine Lacosamide...

disorder. Curry, W. J; Kulling, D. L (1998). "Newer antiepileptic drugs: Gabapentin, lamotrigine, felbamate, topiramate and fosphenytoin". American Family...

bowel or bladder function. Many treatments, including corticosteroids, gabapentin, pregabalin, acupuncture, heat or ice, and spinal manipulation, have limited...

severe allergic reactions due to its strong antihistamine properties. Gabapentin, approved for treatment of seizures and postherpetic neuralgia in adults...