Cholinesterase inhibitors (ChEIs), also known as anti-cholinesterase, are chemicals that prevent the breakdown of the neurotransmitter acetylcholine or...
13 KB (1,107 words) - 21:19, 24 November 2024
with acetylcholin esterase inhibitors and electrical stimulation, the muscle develops trigger points. A cholinesterase inhibitor (or "anticholinesterase")...
17 KB (1,803 words) - 19:04, 26 March 2024
Acetylcholinesterase inhibitors (AChEIs) also often called cholinesterase inhibitors, inhibit the enzyme acetylcholinesterase from breaking down the neurotransmitter...
26 KB (2,387 words) - 03:29, 21 August 2024
Acetylcholine (section Cholinesterase inhibitors)
toxins and venoms produced by plants and animals also contain cholinesterase inhibitors. In clinical use, they are administered in low doses[why?] to...
41 KB (4,382 words) - 05:15, 9 November 2024
crisis may be masked by the concomitant use of atropine along with cholinesterase inhibitor medication in order to prevent side effects. Flaccid paralysis...
7 KB (616 words) - 12:40, 22 May 2024
Dimethoate (category Acetylcholinesterase inhibitors)
organophosphates, dimethoate is an acetylcholinesterase inhibitor which disables cholinesterase, an enzyme essential for central nervous system function...
12 KB (1,065 words) - 11:36, 14 June 2024
discharged from the hospital on 22 September 2020. The OPCW said that a cholinesterase inhibitor from the Novichok group was found in Navalny's blood, urine, skin...
161 KB (14,266 words) - 15:16, 26 October 2024
Tacrine (category Acetylcholinesterase inhibitors)
acetylcholinesterase inhibitor and indirect cholinergic agonist (parasympathomimetic). It was the first centrally acting cholinesterase inhibitor approved for...
9 KB (723 words) - 16:44, 12 July 2024
Rivastigmine (category Acetylcholinesterase inhibitors)
Rivastigmine, a cholinesterase inhibitor, inhibits both butyrylcholinesterase and acetylcholinesterase (unlike donepezil, which selectively inhibits acetylcholinesterase)...
21 KB (1,812 words) - 12:37, 12 October 2024
of mild to moderate dementia of the Alzheimer's type. It is a cholinesterase inhibitor. Benzgalantamine is a prodrug of galantamine. The most common side...
6 KB (202 words) - 20:41, 23 October 2024
announcement, confirming that Navalny had been poisoned with a cholinesterase inhibitor. Ivan Zhdanov, chief of Navalny's Anti-Corruption Foundation, said...
341 KB (29,485 words) - 05:08, 25 November 2024
alkaloid, specifically, a reversible cholinesterase inhibitor CAS 59-99-4 - Neostigmine an acetylcholinesterase inhibitor CAS 317–52–2 - Hexafluronium bromide...
54 KB (5,989 words) - 12:38, 23 November 2024
muscarinic receptors (thus mimicking acetylcholine), or indirectly by inhibiting cholinesterase, promoting acetylcholine release, or other mechanisms. Common...
7 KB (618 words) - 06:38, 29 April 2024
has been used for control of soil-borne nematodes. Aldicarb is a cholinesterase inhibitor, which prevents the breakdown of acetylcholine in the synapse....
4 KB (435 words) - 17:52, 24 January 2024
July 2024. Anti-amyloid drugs also cause brain shrinkage. The cholinesterase inhibitor benzgalantamine was approved by the FDA in July 2024. Specific...
186 KB (19,755 words) - 21:54, 23 November 2024
nature. Naturally occurring aminals Physostigmine,a highly toxic cholinesterase inhibitor found in the Calabar bean. Hodgkinsine, an alkaloid with antiviral...
2 KB (284 words) - 19:10, 19 October 2023
inhibition the substrate and inhibitor cannot bind to the enzyme at the same time.: 134 This usually results from the inhibitor having an affinity for the...
104 KB (11,579 words) - 19:29, 18 September 2024
to suppress sebum production. H1-antihistamines refer to compounds that inhibit the activity of the H1 receptor. Since the H1 receptor exhibits constitutive...
36 KB (3,294 words) - 20:53, 24 November 2024
Neostigmine/glycopyrronium bromide (category Acetylcholinesterase inhibitors)
after surgery. It contains neostigmine as the methylsulfate, a cholinesterase inhibitor, and glycopyrronium bromide, an antimuscarinic agent. Neostigmine/glycopyrronium...
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Ambenonium chloride (category Acetylcholinesterase inhibitors)
Mytelase) is a cholinesterase inhibitor used in the management of myasthenia gravis. It is classified as a reversible cholinesterase inhibitor. Ambenonium...
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Anticholinergic (redirect from Choline inhibitor)
causative agents have been excreted. Reversible acetylcholinesterase inhibitor agents such as physostigmine can be used as an antidote in life-threatening...
25 KB (2,388 words) - 05:24, 21 July 2024
reuptake inhibitor Excitatory amino acid reuptake inhibitor (or glutamate-aspartate reuptake inhibitor) GABA reuptake inhibitor Glycine reuptake inhibitor Monoamine...
19 KB (1,917 words) - 07:07, 23 November 2024
doi:10.1002/ps.4502. PMID 27976502. Gage, J. C. (1 June 1953). "A cholinesterase inhibitor derived from OO -diethyl O - p -nitrophenyl thiophosphate in vivo"...
61 KB (6,918 words) - 15:06, 12 November 2024
chemist. He was known for the synthesis of the first organophosphate cholinesterase inhibitor (tetraethyl pyrophosphate, TEPP). He worked in Adolphe Wurtz's...
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Aldicarb (category Acetylcholinesterase inhibitors)
leafminers, but is primarily used as a nematicide. Aldicarb is a cholinesterase inhibitor which prevents the breakdown of acetylcholine in the synapse. Aldicarb...
12 KB (1,120 words) - 06:02, 19 August 2024
H2 receptor antagonist (redirect from H2 inhibitor)
liver cytochrome P450 (CYP) pathway. To be specific, cimetidine is an inhibitor of the P450 enzymes CYP1A2, CYP2C9, CYP2C19, CYP2D6, CYP2E1, CYP3A4. By...
20 KB (2,234 words) - 18:27, 20 October 2024
Paraoxon (category Acetylcholinesterase inhibitors)
Paraoxon is a parasympathomimetic drug which acts as an cholinesterase inhibitor. It is an organophosphate oxon, and the active metabolite of the insecticide...
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Angiotensin II receptor blocker (redirect from Angiotensin receptor inhibitor)
ACE inhibitor therapy.[citation needed] More recently, they have been used for the treatment of heart failure in patients intolerant of ACE inhibitor therapy...
52 KB (5,172 words) - 06:59, 16 November 2024
Schradan (category Acetylcholinesterase inhibitors)
obsolete organophosphate insecticide. Schradan itself is a weak cholinesterase inhibitor and requires metabolic activation to become active. Dimefox Mipafox...
2 KB (99 words) - 19:34, 12 June 2023
Dopaminergic (section Dopamine reuptake inhibitors)
(June 2024). "A systematic review of the cognitive effects of the COMT inhibitor, tolcapone, in adult humans". CNS Spectr. 29 (3): 166–175. doi:10.1017/S1092852924000130...
28 KB (2,798 words) - 01:21, 21 November 2024