• Thumbnail for Cholinesterase inhibitor
    Cholinesterase inhibitors (ChEIs), also known as anti-cholinesterase, are chemicals that prevent the breakdown of the neurotransmitter acetylcholine or...
    13 KB (1,107 words) - 21:19, 24 November 2024
  • Thumbnail for Cholinesterase
    with acetylcholin esterase inhibitors and electrical stimulation, the muscle develops trigger points. A cholinesterase inhibitor (or "anticholinesterase")...
    17 KB (1,803 words) - 19:04, 26 March 2024
  • Thumbnail for Acetylcholinesterase inhibitor
    Acetylcholinesterase inhibitors (AChEIs) also often called cholinesterase inhibitors, inhibit the enzyme acetylcholinesterase from breaking down the neurotransmitter...
    26 KB (2,387 words) - 03:29, 21 August 2024
  • Thumbnail for Acetylcholine
    toxins and venoms produced by plants and animals also contain cholinesterase inhibitors. In clinical use, they are administered in low doses[why?] to...
    41 KB (4,382 words) - 05:15, 9 November 2024
  • crisis may be masked by the concomitant use of atropine along with cholinesterase inhibitor medication in order to prevent side effects. Flaccid paralysis...
    7 KB (616 words) - 12:40, 22 May 2024
  • Thumbnail for Dimethoate
    Dimethoate (category Acetylcholinesterase inhibitors)
    organophosphates, dimethoate is an acetylcholinesterase inhibitor which disables cholinesterase, an enzyme essential for central nervous system function...
    12 KB (1,065 words) - 11:36, 14 June 2024
  • Thumbnail for Poisoning of Alexei Navalny
    discharged from the hospital on 22 September 2020. The OPCW said that a cholinesterase inhibitor from the Novichok group was found in Navalny's blood, urine, skin...
    161 KB (14,266 words) - 15:16, 26 October 2024
  • Thumbnail for Tacrine
    Tacrine (category Acetylcholinesterase inhibitors)
    acetylcholinesterase inhibitor and indirect cholinergic agonist (parasympathomimetic). It was the first centrally acting cholinesterase inhibitor approved for...
    9 KB (723 words) - 16:44, 12 July 2024
  • Thumbnail for Rivastigmine
    Rivastigmine (category Acetylcholinesterase inhibitors)
    Rivastigmine, a cholinesterase inhibitor, inhibits both butyrylcholinesterase and acetylcholinesterase (unlike donepezil, which selectively inhibits acetylcholinesterase)...
    21 KB (1,812 words) - 12:37, 12 October 2024
  • Thumbnail for Benzgalantamine
    of mild to moderate dementia of the Alzheimer's type. It is a cholinesterase inhibitor. Benzgalantamine is a prodrug of galantamine. The most common side...
    6 KB (202 words) - 20:41, 23 October 2024
  • Thumbnail for Alexei Navalny
    announcement, confirming that Navalny had been poisoned with a cholinesterase inhibitor. Ivan Zhdanov, chief of Navalny's Anti-Corruption Foundation, said...
    341 KB (29,485 words) - 05:08, 25 November 2024
  • alkaloid, specifically, a reversible cholinesterase inhibitor CAS 59-99-4 - Neostigmine an acetylcholinesterase inhibitor CAS 317–52–2 - Hexafluronium bromide...
    54 KB (5,989 words) - 12:38, 23 November 2024
  • muscarinic receptors (thus mimicking acetylcholine), or indirectly by inhibiting cholinesterase, promoting acetylcholine release, or other mechanisms. Common...
    7 KB (618 words) - 06:38, 29 April 2024
  • has been used for control of soil-borne nematodes. Aldicarb is a cholinesterase inhibitor, which prevents the breakdown of acetylcholine in the synapse....
    4 KB (435 words) - 17:52, 24 January 2024
  • Thumbnail for Alzheimer's disease
    July 2024. Anti-amyloid drugs also cause brain shrinkage. The cholinesterase inhibitor benzgalantamine was approved by the FDA in July 2024. Specific...
    186 KB (19,755 words) - 21:54, 23 November 2024
  • Thumbnail for Aminal
    nature. Naturally occurring aminals Physostigmine,a highly toxic cholinesterase inhibitor found in the Calabar bean. Hodgkinsine, an alkaloid with antiviral...
    2 KB (284 words) - 19:10, 19 October 2023
  • Thumbnail for Enzyme inhibitor
    inhibition the substrate and inhibitor cannot bind to the enzyme at the same time.: 134  This usually results from the inhibitor having an affinity for the...
    104 KB (11,579 words) - 19:29, 18 September 2024
  • Thumbnail for Antihistamine
    to suppress sebum production. H1-antihistamines refer to compounds that inhibit the activity of the H1 receptor. Since the H1 receptor exhibits constitutive...
    36 KB (3,294 words) - 20:53, 24 November 2024
  • Neostigmine/glycopyrronium bromide (category Acetylcholinesterase inhibitors)
    after surgery. It contains neostigmine as the methylsulfate, a cholinesterase inhibitor, and glycopyrronium bromide, an antimuscarinic agent. Neostigmine/glycopyrronium...
    5 KB (207 words) - 22:00, 3 November 2024
  • Ambenonium chloride (category Acetylcholinesterase inhibitors)
    Mytelase) is a cholinesterase inhibitor used in the management of myasthenia gravis. It is classified as a reversible cholinesterase inhibitor. Ambenonium...
    4 KB (212 words) - 19:50, 7 September 2024
  • causative agents have been excreted. Reversible acetylcholinesterase inhibitor agents such as physostigmine can be used as an antidote in life-threatening...
    25 KB (2,388 words) - 05:24, 21 July 2024
  • Thumbnail for Reuptake inhibitor
    reuptake inhibitor Excitatory amino acid reuptake inhibitor (or glutamate-aspartate reuptake inhibitor) GABA reuptake inhibitor Glycine reuptake inhibitor Monoamine...
    19 KB (1,917 words) - 07:07, 23 November 2024
  • Thumbnail for Organophosphate
    doi:10.1002/ps.4502. PMID 27976502. Gage, J. C. (1 June 1953). "A cholinesterase inhibitor derived from OO -diethyl O - p -nitrophenyl thiophosphate in vivo"...
    61 KB (6,918 words) - 15:06, 12 November 2024
  • Thumbnail for Philippe de Clermont
    chemist. He was known for the synthesis of the first organophosphate cholinesterase inhibitor (tetraethyl pyrophosphate, TEPP). He worked in Adolphe Wurtz's...
    2 KB (90 words) - 02:32, 14 September 2024
  • Thumbnail for Aldicarb
    Aldicarb (category Acetylcholinesterase inhibitors)
    leafminers, but is primarily used as a nematicide. Aldicarb is a cholinesterase inhibitor which prevents the breakdown of acetylcholine in the synapse. Aldicarb...
    12 KB (1,120 words) - 06:02, 19 August 2024
  • Thumbnail for H2 receptor antagonist
    liver cytochrome P450 (CYP) pathway. To be specific, cimetidine is an inhibitor of the P450 enzymes CYP1A2, CYP2C9, CYP2C19, CYP2D6, CYP2E1, CYP3A4. By...
    20 KB (2,234 words) - 18:27, 20 October 2024
  • Thumbnail for Paraoxon
    Paraoxon (category Acetylcholinesterase inhibitors)
    Paraoxon is a parasympathomimetic drug which acts as an cholinesterase inhibitor. It is an organophosphate oxon, and the active metabolite of the insecticide...
    4 KB (221 words) - 18:23, 29 September 2024
  • Thumbnail for Angiotensin II receptor blocker
    ACE inhibitor therapy.[citation needed] More recently, they have been used for the treatment of heart failure in patients intolerant of ACE inhibitor therapy...
    52 KB (5,172 words) - 06:59, 16 November 2024
  • Thumbnail for Schradan
    Schradan (category Acetylcholinesterase inhibitors)
    obsolete organophosphate insecticide. Schradan itself is a weak cholinesterase inhibitor and requires metabolic activation to become active. Dimefox Mipafox...
    2 KB (99 words) - 19:34, 12 June 2023
  • Thumbnail for Dopaminergic
    (June 2024). "A systematic review of the cognitive effects of the COMT inhibitor, tolcapone, in adult humans". CNS Spectr. 29 (3): 166–175. doi:10.1017/S1092852924000130...
    28 KB (2,798 words) - 01:21, 21 November 2024