A nonsteroidal antiandrogen (NSAA) is an antiandrogen with a nonsteroidal chemical structure. They are typically selective and full or silent antagonists...
17 KB (1,576 words) - 15:57, 24 February 2024
steroidal antiandrogen that has been widely used in the treatment of prostate cancer, but it has largely been replaced by nonsteroidal antiandrogens, which...
158 KB (15,079 words) - 13:02, 1 September 2024
testosterone levels to the female/castrate range. Nonsteroidal antiandrogens are antiandrogens which are nonsteroidal and hence unrelated to steroid hormones in...
232 KB (25,215 words) - 11:40, 1 September 2024
for the same purpose. They are the converse of nonsteroidal antiandrogens (NSAAs), which are antiandrogens that are not steroids and are structurally unrelated...
24 KB (2,340 words) - 08:04, 7 February 2024
progestogens. In addition, it includes both steroidal antiandrogen (SAAs) and nonsteroidal antiandrogen (NSAAs). 17α-Hydroxyprogesterone derivatives Chlormadinone...
5 KB (254 words) - 18:23, 18 September 2023
Comparison of the nonsteroidal antiandrogen (NSAA) bicalutamide with other antiandrogens reveals differences between the medications in terms of efficacy...
85 KB (8,742 words) - 03:27, 16 August 2024
(SGRMTooltip Selective glucocorticoid receptor modulator) Nonsteroidal antiandrogen Nonsteroidal estrogen Edward J. Pavlik (6 December 2012). Estrogens,...
5 KB (381 words) - 23:18, 21 July 2023
Enzalutamide (category Nonsteroidal antiandrogens)
Enzalutamide, sold under the brand name Xtandi, is a nonsteroidal antiandrogen (NSAA) medication which is used in the treatment of prostate cancer. It...
50 KB (4,674 words) - 20:52, 20 August 2024
Apalutamide (category Nonsteroidal antiandrogens)
Apalutamide, sold under the brand name Erleada among others, is a nonsteroidal antiandrogen (NSAA) medication used for the treatment of prostate cancer. It...
36 KB (3,026 words) - 22:35, 16 August 2024
antiandrogens can potentially be used to treat it. As of 2010[update] antiandrogens are small molecules and can be either steroidal or nonsteroidal depending...
42 KB (4,594 words) - 12:17, 24 February 2024
4103/2230-8210.113770. PMC 3743379. PMID 23961495. Gillatt, David (August 2006). "Antiandrogen treatments in locally advanced prostate cancer: are they all the same...
63 KB (6,473 words) - 00:44, 13 June 2024
Thalidomide (category Nonsteroidal antiandrogens)
acts as an antagonist of the androgen receptor and hence is a nonsteroidal antiandrogen of some capacity. In accordance, it can produce gynecomastia and...
76 KB (7,428 words) - 17:54, 30 August 2024
osteoporosis, and benign prostatic hypertrophy (BPH), using the nonsteroidal antiandrogen bicalutamide as a lead compound. Development of andarine for all...
10 KB (958 words) - 17:14, 4 July 2024
Topilutamide (category Nonsteroidal antiandrogens)
known as perfluoroacylamido-arylpropanamides. Topilutamide is a nonsteroidal antiandrogen (NSAA), or an antagonist of the androgen receptor (AR), the biological...
10 KB (762 words) - 22:08, 3 February 2024
structural modification of the arylpropionamide nonsteroidal antiandrogen bicalutamide. They are nonsteroidal arylpropionamides themselves and are close structural...
116 KB (12,935 words) - 04:43, 18 August 2024
The medical uses of bicalutamide, a nonsteroidal antiandrogen (NSAA), include the treatment of androgen-dependent conditions and hormone therapy to block...
133 KB (13,465 words) - 06:08, 1 September 2024
Bicalutamide (category Nonsteroidal antiandrogens)
recommended during treatment. Bicalutamide is a member of the nonsteroidal antiandrogen (NSAA) group of medications. It works by selectively blocking...
217 KB (21,658 words) - 23:36, 31 August 2024
Valproate (category Nonsteroidal antiandrogens)
antagonist of the androgen and progesterone receptors, and hence as a nonsteroidal antiandrogen and antiprogestogen, at concentrations much lower than therapeutic...
93 KB (7,998 words) - 08:10, 27 August 2024
The side effects of bicalutamide, a nonsteroidal antiandrogen (NSAA), including its frequent and rare side effects, have been well-studied and characterized...
140 KB (15,744 words) - 18:51, 1 September 2024
Ketoconazole (category Nonsteroidal antiandrogens)
Ketoconazole, sold under the brand name Nizoral among others, is an antiandrogen, antifungal, and antiglucocorticoid medication used to treat a number...
50 KB (4,379 words) - 13:23, 1 September 2024
Spironolactone (category Steroidal antiandrogens)
Spironolactone, the 5α-reductase inhibitor finasteride, and the nonsteroidal antiandrogen flutamide all appear to have similar effectiveness in the treatment...
181 KB (17,331 words) - 09:05, 1 September 2024
7-8117), or N-(3,5-dimethyl-4-isoxazolylmethyl)phthalimide, is a nonsteroidal antiandrogen (NSAA) structurally related to thalidomide (which also binds to...
7 KB (554 words) - 13:19, 2 March 2024
Rezvilutamide (category Nonsteroidal antiandrogens)
Nonproprietary Name), sold under the brand name Ariane, is a nonsteroidal antiandrogen which is approved for the treatment of prostate cancer in China...
4 KB (181 words) - 20:06, 30 November 2023
RU-58841 (category Nonsteroidal antiandrogens)
RU-58841, also known as PSK-3841 or HMR-3841, is a nonsteroidal antiandrogen (NSAA) which was initially developed in the 1980s by Roussel Uclaf, the French...
6 KB (533 words) - 18:51, 25 October 2023
Pyrilutamide (category Nonsteroidal antiandrogens)
Pyrilutamide (developmental code name KX-826) is a nonsteroidal antiandrogen (NSAA) – specifically, a selective high-affinity silent antagonist of the...
5 KB (258 words) - 17:03, 30 June 2024
Nilutamide (category Nonsteroidal antiandrogens)
Nilutamide, sold under the brand names Nilandron and Anandron, is a nonsteroidal antiandrogen (NSAA) which is used in the treatment of prostate cancer. It has...
52 KB (5,383 words) - 04:40, 11 July 2024
of the pharmacodynamic and pharmacokinetic properties of the nonsteroidal antiandrogen (NSAA) bicalutamide. In terms of pharmacodynamics, bicalutamide...
185 KB (20,418 words) - 12:39, 1 September 2024
Cyproterone acetate (category Antiandrogen esters)
leuprorelin and degarelix, nonsteroidal antiandrogens like flutamide and bicalutamide, the diuretic and steroidal antiandrogen spironolactone, the progestin...
139 KB (13,859 words) - 14:42, 10 July 2024
Darolutamide (category Nonsteroidal antiandrogens)
asthenia, pain in the arms and legs, and rash. Darolutamide is a nonsteroidal antiandrogen (NSAA), and acts as a selective antagonist of the androgen receptor...
42 KB (4,164 words) - 15:13, 25 July 2024
Proxalutamide (category Nonsteroidal antiandrogens)
Proxalutamide (developmental code name GT-0918) is a nonsteroidal antiandrogen (NSAA) – specifically, a selective high-affinity silent antagonist of the...
5 KB (340 words) - 03:30, 19 August 2023