5α-Dihydroethisterone (5α-DHET; developmental code name HE-3562) is an active metabolite of the formerly clinically used but now-discontinued progestin...
13 KB (1,125 words) - 01:45, 18 December 2023
19-Norandrosterone 19-Noretiocholanolone 5α-Dihydronorethandrolone 5α-Dihydronorethisterone 5α-Dihydrolevonorgestrel 5α-Dihydroethisterone Kicman AT (June 2008). "Pharmacology...
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17α-Allyl-19-nortestosterone 20α-Dihydrodydrogesterone 5α-Dihydrolevonorgestrel 5α-Dihydroethisterone Ethinylandrostenediol Hydroxytibolones 3α-Hydroxytibolone...
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17α-Ethynyl-3α-androstanediol (redirect from 17α-ethynyl-5α-androstane-3α,17β-diol)
its mechanism of action is not well-characterized. It produces 5α-dihydroethisterone (5α-dihydro-17α-ethynyltestosterone), a ligand of several steroid...
6 KB (377 words) - 20:25, 10 February 2024
5α-Dihydroprogesterone (5α-DHP, allopregnanedione, or 5α-pregnane-3,20-dione) is an endogenous progestogen and neurosteroid that is synthesized from progesterone...
10 KB (909 words) - 23:12, 9 November 2023
17α-Ethynyl-3β-androstanediol (redirect from 17α-ethynyl-5α-androstane-3β,17β-diol)
17α-Ethynyl-3β-androstanediol may produce 17α-ethynyl-3α-androstanediol and 5α-dihydroethisterone (5α-dihydro-17α-ethynyltestosterone) as active metabolites in vivo...
6 KB (412 words) - 07:42, 23 May 2023
5α-Dihydronormethandrone (5α-DHNMT; developmental code name RU-575), also known as 17α-methyl-4,5α-dihydro-19-nortestosterone or as 17α-methyl-5α-estran-17β-ol-3-one...
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Dihydrotestosterone (redirect from 5α-Dihydrotestosterone)
Dihydrotestosterone (DHT, 5α-dihydrotestosterone, 5α-DHT, androstanolone or stanolone) is an endogenous androgen sex steroid and hormone primarily involved...
67 KB (6,821 words) - 20:22, 2 August 2024
activity of high doses of levonorgestrel. 5α-Dihydronorethisterone 5α-Dihydroethisterone 5α-Dihydronandrolone 5α-Dihydronormethandrone Kuhl H (2005). "Pharmacology...
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Androstane (redirect from 5α-androstane)
can exist as either of two isomers, known as 5α-androstane and 5β-androstane. 5α-Androstane 5β-Androstane 5α-Androstane is reported to be effective as an...
3 KB (126 words) - 09:16, 13 December 2023
5α-DHNET has been proposed as a potential therapeutic agent in the treatment of estrogen receptor (ER)-positive breast cancer. 5α-Dihydroethisterone...
9 KB (772 words) - 17:43, 11 November 2023
Danazol 9 8 ? <0.2a ? 40 10 Ethisterone 35 <1 <1 <1b <1 92–121 0.33 5α-Dihydroethisterone 12 38–100c 4 120b ? 100 ? Notes: Values are percentages (%). Reference...
46 KB (3,954 words) - 04:46, 8 April 2024
where androstenedione is converted into 5α-dihydrotestosterone (DHT) and testosterone (T) in male and into 5α-dihydroandrostenedione (DHA) in females...
19 KB (1,899 words) - 15:35, 24 January 2024
groups, respectively. For example, 5α-pregnane-3α,17α-diol-20-one has a hydrogen atom at the 5α position (hence the "5α-" prefix), two hydroxy groups (-OH)...
83 KB (8,473 words) - 20:30, 10 October 2024
5α-Dihydronorethandrolone (5α-DHNED), also known as 17α-ethyl-4,5α-dihydro-19-nortestosterone or as 17α-ethyl-5α-estran-17β-ol-3-one, is an androgen/anabolic...
3 KB (126 words) - 17:43, 11 November 2023
5α-dihydroprogesterone (5α-DHP), 5β-dihydroprogesterone (5β-DHP) (very weak), 3β-dihydroprogesterone (3β-DHP), 11-deoxycorticosterone (DOC), and 5α...
16 KB (1,567 words) - 01:04, 8 October 2024
hepatotoxicity. Drostanolone, also known as 2α-methyl-5α-dihydrotestosterone (2α-methyl-DHT) or as 2α-methyl-5α-androstan-17β-ol-3-one, is a synthetic androstane...
11 KB (857 words) - 21:07, 29 February 2024
such, it was not further developed. Zanoterone was derived from 5α-dihydroethisterone (5α-dihydro-17α-ethynyltestosterone). It is an antagonist of the androgen...
7 KB (564 words) - 23:58, 8 December 2023
ethinylestradiol (17α-ethynylestradiol). 5α-Dihydroethisterone (5α-dihydro-17α-ethynyltestosterone), formed by 5α-reductase, is an active metabolite of ethisterone...
31 KB (2,863 words) - 17:44, 11 November 2023
dihydroboldenone, is a synthetic anabolic–androgenic steroid (AAS) and a 5α-reduced derivative of boldenone (Δ1-testosterone). It differs from testosterone...
5 KB (400 words) - 19:27, 25 June 2024
Dihydrodeoxycorticosterone (redirect from 5α-Dihydrodeoxycorticosterone)
5α-Dihydrodeoxycorticosterone (abbreviated as DHDOC), also known as 21-hydroxy-5α-pregnan-20-one, is an endogenous progestogen and neurosteroid. It is...
3 KB (147 words) - 20:19, 30 April 2023
3α-Androstanediol (redirect from 3α,5α-Androstanediol)
3α-Androstanediol also known as 5α-androstane-3α,17β-diol and sometimes shortened in the literature to 3α-diol, is an endogenous steroid hormone and neurosteroid...
10 KB (885 words) - 19:14, 8 April 2024
17β-dihydroxy-5α-androstane and 3α,17β-dihydroxy-5α-androstane) Androstanedione (5α-androstan-3,17-dione) 1-Androstenediol (3α,17β-dihydroxy-5α-androst-1-ene)...
13 KB (1,375 words) - 00:13, 1 September 2024
orally active. It occurs as an important active metabolite of oral TU. The 5α-reductase inhibitor finasteride in combination with oral TU has no effect...
7 KB (529 words) - 15:19, 12 May 2024
Methasterone, also known as 2α,17α-dimethyl-5α-dihydrotestosterone (2α,17α-dimethyl-DHT) or as 2α,17α-dimethyl-5α-androstan-17β-ol-3-one, is a synthetic androstane...
11 KB (1,015 words) - 07:25, 21 May 2024
As oxandrolone is already a 5α-reduced steroid (has a single bond between carbons 4 and 5), it is not a substrate for the 5α-reductase enzyme, hence is...
47 KB (4,522 words) - 20:23, 12 October 2024
Norethisterone (category 5α-Reductase inhibitors)
represented by 5α- and 5β-reduced NET (5α-NET or 5β-NET) and by 3α- and 3β-hydrogenated 5α-NET and 5β-NET, leading to 3α,5α-NET, 3β,5α-NET, 3α,5β-NET...
95 KB (9,417 words) - 16:47, 15 October 2024
percent of testosterone enanthate will be converted to 5α-dihydrotestosterone in normal men. 5α-Dihydrotestosterone (DHT) can promote masculine characteristics...
26 KB (2,246 words) - 18:23, 12 October 2024
Androstanedione (redirect from 5α-androstanedione)
Androstanedione, also known as 5α-androstanedione or as 5α-androstane-3,17-dione, is a naturally occurring androstane (5α-androstane) steroid and an endogenous...
4 KB (211 words) - 17:41, 11 November 2023
Epiandrosterone (category 5α-Reduced steroid metabolites)
or isoandrosterone, also known as 3β-androsterone, 3β-hydroxy-5α-androstan-17-one, or 5α-androstan-3β-ol-17-one, is a steroid hormone with weak androgenic...
7 KB (606 words) - 17:44, 11 November 2023