The beta-3 adrenergic receptor (β3-adrenoceptor), also known as ADRB3, is a beta-adrenergic receptor, and also denotes the human gene encoding it. Actions...
17 KB (2,039 words) - 09:45, 7 October 2023
The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...
33 KB (3,420 words) - 14:42, 6 November 2024
The beta-1 adrenergic receptor (β1 adrenoceptor), also known as ADRB1, can refer to either the protein-encoding gene (gene ADRB1) or one of the four adrenergic...
31 KB (3,742 words) - 16:12, 25 October 2024
The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline)...
33 KB (2,982 words) - 11:42, 7 August 2024
Beta adrenergic agonists or beta agonists are medications that relax muscles of the airways, causing widening of the airways and resulting in easier breathing...
10 KB (851 words) - 21:05, 24 November 2024
types of β-adrenergic receptors and others are selective for one of the three known types of beta receptors, designated β1, β2 and β3 receptors.: 153 β1-adrenergic...
75 KB (7,463 words) - 18:51, 13 November 2024
The β3 (beta 3) adrenergic receptor agonist or β3-adrenoceptor agonist, also known as β3-AR agonist, are a class of medicine that bind selectively to...
21 KB (2,189 words) - 16:52, 12 October 2024
A Beta-3 adrenergic antagonist (β3-adrenoceptor antagonist) is an adrenergic antagonist which blocks the Beta-3 adrenergic receptors of cells, with either...
1 KB (111 words) - 06:08, 1 May 2023
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are subdivided...
16 KB (1,528 words) - 10:28, 23 June 2024
Beta2-adrenergic agonists, also known as adrenergic β2 receptor agonists, are a class of drugs that act on the β2 adrenergic receptor. Like other β adrenergic...
18 KB (1,703 words) - 06:18, 17 March 2024
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the human gene encoding it. α2...
12 KB (1,303 words) - 04:16, 13 August 2024
The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...
25 KB (2,231 words) - 17:54, 18 September 2024
into two groups. The first group of receptors are the beta (β) adrenergic receptors. There are β1, β2, and β3 receptors. The second group contains the alpha...
15 KB (1,535 words) - 19:07, 2 August 2024
enzymology, a beta-adrenergic-receptor kinase (EC 2.7.11.15) is an enzyme that catalyzes the chemical reaction: ATP + [beta-adrenergic receptor] ⇌ {\displaystyle...
4 KB (381 words) - 18:21, 23 August 2024
G-protein-coupled receptor kinase 2 (GRK2) is an enzyme that in humans is encoded by the ADRBK1 gene. GRK2 was initially called Beta-adrenergic receptor kinase (βARK...
14 KB (1,637 words) - 11:17, 19 June 2022
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of adrenergic receptors are: α1, α2...
7 KB (757 words) - 22:26, 10 September 2024
Vibegron (category Beta3-adrenergic agonists)
the treatment of overactive bladder. Vibegron is a selective beta-3 adrenergic receptor agonist. The most common side effects include headache, urinary...
25 KB (2,260 words) - 01:26, 2 September 2024
Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has...
13 KB (1,359 words) - 20:52, 24 November 2024
A Beta-2 adrenergic antagonist (β2-adrenoceptor antagonist) is an adrenergic antagonist which blocks the beta-2 adrenergic receptors of cells, with either...
1 KB (104 words) - 20:58, 12 August 2023
Propranolol (redirect from Beta-Neg)
considered to be safe. It is a non-selective beta blocker which works by blocking β-adrenergic receptors. Propranolol was patented in 1962 and approved...
51 KB (4,662 words) - 21:24, 25 November 2024
Adrenergic receptor autoantibodies The adrenergic receptors (or adrenoreceptors) are a class of cell membrane-bound protein receptors throughout the body...
15 KB (1,636 words) - 03:12, 2 November 2024
epinephrine. These chemicals will act on adrenergic receptors, with subtypes Alpha-1, Alpha-2, Beta-1, Beta-2, Beta-3, which ultimately allow the body to trigger...
38 KB (3,642 words) - 16:12, 19 November 2024
appears to enhance lipolysis in mice by upregulating beta-3 adrenergic receptors. Beta-3 adrenergic receptor knockout mice are unresponsive to the lipolytic...
5 KB (312 words) - 23:47, 17 August 2024
G-protein-coupled receptor kinase 3 (GRK3) is an enzyme that in humans is encoded by the ADRBK2 gene. GRK3 was initially called Beta-adrenergic receptor kinase 2...
16 KB (2,012 words) - 14:01, 20 January 2024
Sympatholytic (redirect from Adrenergic neurone blockers)
norepinephrine. They are primarily postsynaptic adrenergic receptor antagonists (alpha and beta adrenergic receptor antagonists, or "blockers"), inhibiting the...
11 KB (1,303 words) - 21:40, 3 December 2023
Sympathomimetic drug (redirect from Adrenergic agent)
have greater beta adrenergic receptor activity, but if the substituent is not bulky, then it will favor the alpha adrenergic receptors. Direct stimulation...
9 KB (891 words) - 19:06, 3 September 2024
Adrenergic means "working on adrenaline (epinephrine) or noradrenaline (norepinephrine)" (or on their receptors). When not further qualified, it is usually...
3 KB (286 words) - 18:10, 25 July 2024
β1-Adrenergic receptor agonists, also known as beta-1 agonists, are a class of drugs that bind selectively to the β1-adrenergic receptor. As a result...
4 KB (322 words) - 00:48, 23 July 2024
signalling roles in their own right. Arrestin beta 2, like arrestin beta 1, was shown to inhibit beta-adrenergic receptor function in vitro. It is expressed at...
17 KB (1,965 words) - 19:41, 26 October 2024
β adrenergic receptor antagonists (also called beta-blockers or β-blockers) were initially developed in the 1960s, for the treatment of angina pectoris...
36 KB (4,063 words) - 07:02, 11 December 2023