Nilutamide, sold under the brand names Nilandron and Anandron, is a nonsteroidal antiandrogen (NSAA) which is used in the treatment of prostate cancer...
52 KB (5,388 words) - 17:34, 11 November 2024
parameters. Relative to the other first-generation NSAAs, flutamide and nilutamide, bicalutamide shows improved potency, efficacy, tolerability, and safety...
85 KB (8,727 words) - 01:24, 2 September 2024
or other first-generation NSAAs (i.e., flutamide and nilutamide). A massive overdose of nilutamide (13 grams, or 43 times the normal maximum 300 mg/day...
217 KB (21,648 words) - 17:51, 11 November 2024
different side-chain. These compounds are similar in chemical structure to nilutamide, which is related to flutamide, bicalutamide, and enzalutamide, all of...
6 KB (533 words) - 18:51, 25 October 2023
largely replaced the earlier nonsteroidal antiandrogens flutamide and nilutamide, which are now little used. The earlier androgen synthesis inhibitors...
159 KB (15,083 words) - 17:38, 19 November 2024
Toremifene L02BA03 Fulvestrant L02BA04 Elacestrant L02BB01 Flutamide L02BB02 Nilutamide L02BB03 Bicalutamide L02BB04 Enzalutamide L02BB05 Apalutamide L02BB06...
2 KB (239 words) - 00:26, 31 December 2023
associated side effect of certain drugs such as disulfiram, metronidazole, or nilutamide. Skin flushing and nasal congestion are the most common symptoms of intolerance...
20 KB (1,912 words) - 22:19, 23 May 2024
Cyanonilutamide (redirect from Cyano-nilutamide)
shows significant antiandrogenic activity in animals. 5N-Bicalutamide Nilutamide RU-56187 RU-58642 RU-59063 Gryder BE, Akbashev MJ, Rood MK, Raftery ED...
3 KB (163 words) - 21:36, 22 January 2023
nilestriol (INN) nilotinib (USAN) nilprazole (INN) Nilstat niludipine (INN) nilutamide (INN) nilvadipine (INN) nimazone (INN) Nimbex nimesulide (INN) nimetazepam...
9 KB (417 words) - 07:03, 15 August 2024
level ATC chemical subgroup (L02BG Aromatase inhibitors) Flutamide and nilutamide are alternatives Goserelin and triptorelin are alternatives Prednisone...
67 KB (4,835 words) - 08:21, 11 November 2024
treatment of prostate cancer. In 1995, bicalutamide was approved, and nilutamide followed a year later. The AR belongs to the steroid receptor subfamily...
42 KB (4,594 words) - 12:34, 28 September 2024
comparison to first-generation NSAAs such as bicalutamide, flutamide, and nilutamide. Also, unlike with the first-generation NSAAs, there has been no evidence...
50 KB (4,689 words) - 17:13, 11 November 2024
phosphate; antiandrogens such as nonsteroidal antiandrogens like flutamide, nilutamide, and bicalutamide; and androgen synthesis inhibitors such as ketoconazole...
24 KB (2,462 words) - 23:13, 21 November 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
9 KB (376 words) - 17:45, 11 November 2023
antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol (pentetrazol) Phenylsilatrane Picrotoxin...
37 KB (3,825 words) - 21:25, 7 October 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
149 KB (15,703 words) - 16:01, 5 November 2024
antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol (pentetrazol) Phenylsilatrane Picrotoxin...
53 KB (5,741 words) - 00:23, 23 October 2024
antiandrogen (SAA) cyproterone acetate (CPA) and the NSAAs flutamide and nilutamide, bicalutamide shows an improved profile of effectiveness, tolerability...
134 KB (13,465 words) - 11:13, 2 November 2024
antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol (pentetrazol) Phenylsilatrane Picrotoxin...
89 KB (9,448 words) - 10:19, 5 October 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
7 KB (505 words) - 09:37, 4 November 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
29 KB (3,167 words) - 11:40, 22 November 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
23 KB (1,906 words) - 08:25, 12 July 2024
a nonsteroidal antiandrogen (NSAA) related to the NSAAs flutamide and nilutamide (RU-23908) and was developed by Roussel Uclaf but was never marketed....
4 KB (212 words) - 12:12, 29 September 2024
antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide) Oenanthotoxin Pentylenetetrazol (pentetrazol) Phenylsilatrane Picrotoxin...
37 KB (3,619 words) - 01:04, 1 September 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
74 KB (7,439 words) - 22:39, 25 October 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
209 KB (21,565 words) - 19:39, 16 November 2024
Bicalutamide Cimetidine Darolutamide Enzalutamide Flutamide Ketoconazole Nilutamide Seviteronel† Topilutamide (fluridil) Steroidogenesis inhibitors Antigonadotropins...
181 KB (17,370 words) - 08:34, 11 November 2024
N-Butylbenzenesulfonamide N-Desmethylapalutamide N-Desmethylenzalutamide Nilutamide ONC1-13B Pentomone PF-998425 Phenothrin Prochloraz Procymidone Proxalutamide...
83 KB (8,523 words) - 03:36, 18 November 2024
first-generation NSAA nilutamide and by extension from flutamide. Chemical structures of apalutamide and its predecessors Flutamide Nilutamide RU-59063 Enzalutamide...
36 KB (3,026 words) - 22:35, 16 August 2024
also acting as AR antagonists. First-generation Bicalutamide Flutamide Nilutamide Second-generation Apalutamide Darolutamide Enzalutamide Proxalutamide...
5 KB (254 words) - 18:23, 18 September 2023