field of molecular biology, the peroxisome proliferator–activated receptors (PPARs) are a group of nuclear receptor proteins that function as transcription...
18 KB (1,902 words) - 09:05, 2 October 2024
Peroxisome proliferator-activated receptor gamma (PPAR-γ or PPARG), also known as the glitazone reverse insulin resistance receptor, or NR1C3 (nuclear...
19 KB (2,091 words) - 05:22, 13 July 2024
proliferator-activated receptor delta and peroxisome proliferator-activated receptor gamma, PPAR-alpha is part of the subfamily of peroxisome proliferator-activated receptors...
22 KB (2,567 words) - 22:11, 22 August 2024
Peroxisome proliferator-activated receptor delta (PPAR-delta), or (PPAR-beta), also known as Nuclear hormone receptor 1 (NUC1) is a nuclear receptor that...
18 KB (1,963 words) - 18:29, 24 August 2024
PPAR agonist (redirect from Peroxisome proliferator-activated receptor agonist)
PPAR agonists are drugs which act upon the peroxisome proliferator-activated receptor. They are used for the treatment of symptoms of the metabolic syndrome...
9 KB (1,045 words) - 10:21, 18 July 2024
Telmisartan (category Angiotensin II receptor antagonists)
system, telmisartan acts as a selective modulator of peroxisome proliferator-activated receptor gamma (PPAR-γ), a central regulator of insulin and glucose...
14 KB (1,192 words) - 05:32, 13 September 2024
very-low-density lipoprotein (VLDL). Acadesine GFT505 GW0742 Irisin Peroxisome proliferator-activated receptor Sodelglitazar SR9009 Koh B (2013-03-22). "Anti-doping...
20 KB (1,953 words) - 04:39, 4 August 2024
Peroxisome proliferator-activated receptor gamma coactivator 1-alpha (PGC-1α) is a protein that in humans is encoded by the PPARGC1A gene. PPARGC1A is...
31 KB (3,777 words) - 20:49, 25 September 2024
(January 2004). "Peroxisome proliferator-activated receptor-gamma coactivator 1alpha (PGC-1alpha) regulates triglyceride metabolism by activation of the nuclear...
17 KB (1,945 words) - 06:08, 25 July 2024
increased risk of rhabdomyolysis. Fibrates stimulate peroxisome proliferator activated receptor (PPAR) alpha, which controls the expression of gene products...
10 KB (1,091 words) - 19:45, 8 September 2024
TZDs act by activating PPARs (peroxisome proliferator-activated receptors), a group of nuclear receptors, specific for PPARγ (PPAR-gamma, PPARG). They...
20 KB (2,167 words) - 15:13, 20 September 2024
Notopterygium incisum--new selective partial agonists of peroxisome proliferator-activated receptor-gamma". PLOS ONE. 8 (4): e61755. Bibcode:2013PLoSO...861755A...
4 KB (429 words) - 04:01, 14 February 2024
Phagocytosis (section Initiating receptors)
apoptotic cells in mice with macrophage peroxisome proliferator-activated receptor gamma or retinoid X receptor alpha deficiency". Journal of Immunology...
22 KB (2,451 words) - 14:47, 31 August 2024
Pioglitazone selectively stimulates the nuclear receptor peroxisome proliferator-activated receptor gamma (PPAR-γ) and to a lesser extent PPAR-α. It modulates...
28 KB (2,663 words) - 03:58, 30 September 2024
triggering the activation of AMP-activated protein kinase (AMPK) which subsequently phosphorylates peroxisome proliferator-activated receptor gamma coactivator-1α...
81 KB (10,469 words) - 11:20, 28 September 2024
and obovatol. Magnolol and honokiol activate the nuclear receptor peroxisome proliferator-activated receptor gamma. White or Yulan magnolia (subgenus Yulania)...
47 KB (5,056 words) - 22:13, 14 September 2024
PPAR agonist at the subtypes α (alpha) and γ (gamma) of the peroxisome proliferator-activated receptor (PPAR). Agonist action on PPARα lowers high blood...
9 KB (746 words) - 07:01, 29 May 2024
metabolite GFT1007 are peroxisome proliferator-activated receptor (PPAR) agonists, both of which activate PPAR-alpha, PPAR-gamma, and PPAR-delta in vitro...
13 KB (782 words) - 22:24, 30 September 2024
NFKB1, PCAF, PPARGC1A, Peroxisome proliferator-activated receptor alpha, SNW1, STAT3, STAT6, TRIP4, and Thyroid hormone receptor beta. GRCh38: Ensembl...
15 KB (1,725 words) - 17:17, 1 July 2024
lipolysis. It does so by activating peroxisome proliferator-activated receptor alpha (PPARα) 'transcription factor ligand', a receptor that is involved in...
12 KB (950 words) - 06:13, 1 April 2024
"Estrogen-related receptor-gamma and peroxisome proliferator-activated receptor-gamma coactivator-1alpha regulate estrogen-related receptor-alpha gene expression...
10 KB (1,243 words) - 09:39, 12 October 2023
ester. It lowers lipid levels by activating peroxisome proliferator-activated receptor alpha (PPARα). PPARα activates lipoprotein lipase and reduces apoprotein...
26 KB (2,514 words) - 21:09, 28 September 2024
proposed to be the peroxisome proliferator-activated receptor alpha (PPAR-α). PEA also has affinity to cannabinoid-like G-coupled receptors GPR55 and GPR119...
47 KB (5,039 words) - 04:14, 20 September 2024
Pemafibrate, sold under the brand namd Parmodia, is a peroxisome proliferator-activated receptor alpha (PPARα) agonist. It is developed and marketed by...
4 KB (91 words) - 16:40, 23 September 2024
diabetic human coronary artery endothelial cells through peroxisome proliferator-activated receptor gamma". Molecular and Cellular Endocrinology. 412: 320–329...
27 KB (2,969 words) - 23:05, 2 September 2024
alpha, Estrogen receptor beta, Glucocorticoid receptor, IKBKG, IKK2, Peroxisome proliferator-activated receptor gamma, and Retinoid X receptor alpha. GRCh38:...
21 KB (2,438 words) - 21:40, 11 July 2024
"15-deoxy-delta12,14-prostaglandin J2, a specific ligand for peroxisome proliferator-activated receptor-gamma, induces neuronal apoptosis". NeuroReport. 12 (4):...
23 KB (3,059 words) - 16:19, 5 November 2023
diabetic human coronary artery endothelial cells through peroxisome proliferator-activated receptor gamma". Molecular and Cellular Endocrinology. 412: 320–329...
100 KB (11,155 words) - 18:45, 24 August 2024
Roberts-Thomson SJ (July 2004). "Effect of the peroxisome proliferator-activated receptor beta activator GW0742 in rat cultured cerebellar granule neurons"...
9 KB (827 words) - 19:19, 6 May 2024
Arachidonic acid (section PLA2 activation)
arachidonic acid. Receptors that activate this pathway include: A1 receptor D2 receptor α2 adrenergic receptor 5-HT1 receptor PLC may also be activated by MAP kinase...
21 KB (1,899 words) - 18:33, 30 September 2024