Rimonabant (also known as SR141716; trade names Acomplia, Zimulti) is an anorectic antiobesity drug approved in Europe in 2006 but was withdrawn worldwide...
14 KB (1,176 words) - 06:15, 27 November 2024
Cannabinoid receptor antagonist (section Rimonabant)
receptor antagonists. The first CBR inverse agonist, rimonabant, was described in 1994. Rimonabant blocks the CB1 receptor selectively and has been shown...
41 KB (4,204 words) - 03:27, 9 October 2024
at the CB1 cannabinoid receptor. AM-251 is structurally very close to rimonabant; both are biarylpyrazole cannabinoid receptor antagonists. In AM-251,...
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oxaloacetate supplements had no effect on lifespan in healthy laboratory mice. Rimonabant (Acomplia) is an anti-obesity drug initially approved for use in the European...
23 KB (2,847 words) - 16:57, 24 November 2024
cannabis), increased appetite. However, some drugs in this class such as rimonabant were withdrawn or ceased development to concerns about mental health and...
54 KB (5,046 words) - 17:44, 3 December 2024
drugs that were ever approved by the FDA. Some of them (lumiracoxib, rimonabant, tolrestat, ximelagatran and ximelidine, for example) were approved to...
45 KB (1,903 words) - 16:52, 9 October 2024
The antihypertensive effect of spilanthol was blocked by CB1 antagonist rimonabant and TRPV1 antagonist capsazepine, suggesting spilanthol mediates some...
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seen with an antagonist. An example is the cannabinoid inverse agonist rimonabant. A superagonist is a term used by some to identify a compound that is...
14 KB (1,622 words) - 03:21, 4 September 2024
Protriptyline Proparacaine Quetiapine Ramelteon Rasagiline Reboxetine Ribavirin Rimonabant Risperidone Rivastigmine Rofecoxib Ropinirole Rotigotine Rufinamide Selegiline...
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Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
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depression, and thoughts of suicide in patients treated with the now-withdrawn rimonabant, another CB1 antagonist that was also under development by Sanofi-Aventis...
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O-1918 O-2050 O-2654 Otenabant (CP-945,598) PF-514273 PipISB PSB-SB-487 Rimonabant (SR141716) Rosonabant (E-6776) SR-144,528 Surinabant (SR147778) Taranabant...
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including flunarizine, mefloquine, and efavirenz. Another notable agent is rimonabant, a cannabinoid receptor antagonist marketed as an anti-obesity agent which...
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adverse cardiovascular risk profile. Similarly, the appetite suppressant rimonabant (a cannabinoid receptor antagonist) had to be withdrawn when it was linked...
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adenosine A1 receptor agonists. Cannabinoid CB1 receptor antagonists like rimonabant, drinabant, and surinabant have been found to block or reduce the psychoactive...
36 KB (3,962 words) - 07:55, 26 November 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
34 KB (3,188 words) - 04:03, 23 November 2024
Federal Analogue Act Hexahydrocannabivarin Medical cannabis Parahexyl Rimonabant (synthetic CB1 antagonist) Tetrahydrocannabiorcol (Δ9-THCC, (C1)-Δ9-THC)...
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Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
176 KB (16,457 words) - 17:54, 2 January 2025
UR-144 WIN 55,212-2 Yangonin Inverse agonists AM-251 INV-202 Monlunabant Rimonabant Surinabant Taranabant TM-38837 Zevaquenabant Antagonists AM-6545 Cannabidiol...
122 KB (12,163 words) - 14:36, 3 January 2025
selective for the CB1 receptor over CB2, than the more commonly used ligand rimonabant, with a Ki at CB1 of 350fM (i.e. 0.00035nM) and a selectivity of over...
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discontinued following the problems seen during clinical use of the similar drug rimonabant. Cannabinoid receptor antagonist Kim MA, Yun H, Kwak H, Kim J, Lee J (2008)...
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Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
125 KB (11,614 words) - 10:24, 3 January 2025
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
116 KB (11,946 words) - 11:38, 30 December 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
143 KB (13,847 words) - 13:44, 10 December 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
51 KB (4,625 words) - 01:01, 25 December 2024
UR-144 WIN 55,212-2 Yangonin Inverse agonists AM-251 INV-202 Monlunabant Rimonabant Surinabant Taranabant TM-38837 Zevaquenabant Antagonists AM-6545 Cannabidiol...
72 KB (8,093 words) - 23:02, 30 December 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
28 KB (2,386 words) - 06:04, 1 December 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
53 KB (5,956 words) - 21:49, 19 December 2024
Naloxone Naltrexazone Naltrexonazine Naltrexone Naltrindole Naringenin Noribogaine Oxilorphan Pawhuskin A Rimonabant Quadazocine Samidorphan Taxifolin...
55 KB (4,903 words) - 23:55, 2 January 2025
naltrexone A08AB01 Orlistat QA08AB90 Mitratapide QA08AB91 Dirlotapide A08AX01 Rimonabant Diet products are in the ATC group V06A. "ATC (Anatomical Therapeutic...
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