The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline)...
33 KB (2,982 words) - 11:42, 7 August 2024
The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...
25 KB (2,231 words) - 17:54, 18 September 2024
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are subdivided...
16 KB (1,528 words) - 10:28, 23 June 2024
The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...
33 KB (3,418 words) - 12:27, 19 September 2024
Beta blocker (redirect from Beta-adrenergic receptor antagonists)
and β3 receptors.: 153 β1-adrenergic receptors are located mainly in the heart and in the kidneys. β2-adrenergic receptors are located mainly in the lungs...
75 KB (7,463 words) - 04:42, 2 October 2024
adrenergic receptor (β1 adrenoceptor), also known as ADRB1, can refer to either the protein-encoding gene (gene ADRB1) or one of the four adrenergic receptors...
31 KB (3,742 words) - 18:01, 29 August 2024
Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has...
13 KB (1,360 words) - 22:27, 10 September 2024
alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic receptor, is an alpha-1 adrenergic receptor...
11 KB (1,360 words) - 10:20, 23 June 2024
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of adrenergic receptors are: α1, α2...
7 KB (757 words) - 22:26, 10 September 2024
The beta-3 adrenergic receptor (β3-adrenoceptor), also known as ADRB3, is a beta-adrenergic receptor, and also denotes the human gene encoding it. Actions...
17 KB (2,039 words) - 09:45, 7 October 2023
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the human gene encoding it. α2...
12 KB (1,303 words) - 04:16, 13 August 2024
Beta2-adrenergic agonists, also known as adrenergic β2 receptor agonists, are a class of drugs that act on the β2 adrenergic receptor. Like other β adrenergic...
18 KB (1,703 words) - 06:18, 17 March 2024
Adrenergic means "working on adrenaline (epinephrine) or noradrenaline (norepinephrine)" (or on their receptors). When not further qualified, it is usually...
3 KB (286 words) - 18:10, 25 July 2024
Adrenergic receptor autoantibodies The adrenergic receptors (or adrenoreceptors) are a class of cell membrane-bound protein receptors throughout the body...
15 KB (1,636 words) - 02:22, 19 September 2024
The alpha-2B adrenergic receptor (α2B adrenoceptor), is a G-protein coupled receptor. It is a subtype of the adrenergic receptor family. The human gene...
15 KB (1,754 words) - 20:51, 13 August 2023
The alpha-2C adrenergic receptor (α2C adrenoceptor), also known as ADRA2C, is an alpha-2 adrenergic receptor, and also denotes the human gene encoding...
13 KB (1,541 words) - 00:52, 27 September 2024
Pharmacology of Adrenergic Receptors". Meyers, D.S.; Skwish, S.; Dickinson, K.E.; Kienzle, B.; Arbeeny, C.M. (Feb 1997). "Beta 3-adrenergic receptor-mediated...
9 KB (805 words) - 07:26, 20 August 2024
An adrenergic antagonist is a drug that inhibits the function of adrenergic receptors. There are five adrenergic receptors, which are divided into two...
15 KB (1,535 words) - 19:07, 2 August 2024
The alpha-1B adrenergic receptor (α1B-adrenoreceptor), also known as ADRA1B, is an alpha-1 adrenergic receptor, and also denotes the human gene encoding...
11 KB (1,333 words) - 02:33, 18 October 2022
Antihypertensive (redirect from Alpha-2 adrenergic receptor agonist)
Beta-blockers can block beta-1 adrenergic receptors and/or beta-2 adrenergic receptors. Those that block beta-1-adrenergic receptors prevent the binding of endogenous...
56 KB (6,325 words) - 18:29, 22 September 2024
Selective androgen receptor modulators (SARMs) are a class of drugs that selectively activate the androgen receptor in specific tissues, promoting muscle...
74 KB (6,763 words) - 03:02, 16 September 2024
of β2-adrenergic receptor (β2AR) with a diffusible ligand brought surprising results because it revealed quite a different shape of the receptor extracellular...
82 KB (9,384 words) - 16:34, 5 September 2024
adrenergic receptor agonist or β3-adrenoceptor agonist, also known as β3-AR agonist, are a class of medicine that bind selectively to β3-adrenergic receptors...
21 KB (2,188 words) - 03:36, 20 October 2023
Sympathomimetic drug (redirect from Adrenergic agent)
direct-acting (direct interaction between drug and receptor), such as α-adrenergic agonists, β-adrenergic agonists, and dopaminergic agonists; or indirect-acting...
9 KB (891 words) - 19:06, 3 September 2024
Alpha blocker (redirect from Alpha-adrenergic blocker)
are a class of pharmacological agents that act as antagonists on α-adrenergic receptors (α-adrenoceptors). Historically, alpha-blockers were used as a tool...
34 KB (3,215 words) - 03:11, 10 September 2024
Sympatholytic (redirect from Adrenergic neurone blockers)
pathways of adrenergic receptors. However, there are exceptions: clonidine is an adrenergic agonist at the α2 receptor; since this receptor is located...
11 KB (1,303 words) - 21:40, 3 December 2023
The alpha-1D adrenergic receptor (α1D adrenoreceptor), also known as ADRA1D, is an alpha-1 adrenergic receptor, and also denotes the human gene encoding...
10 KB (1,214 words) - 05:09, 20 September 2024
β1-adrenergic receptor (Ki = 0.24–0.43 nM), β2-adrenergic receptor (Ki = 0.19–0.25 nM), α1-adrenergic receptor (Ki = 3.4 nM), α2-adrenergic receptor (Ki...
33 KB (2,908 words) - 03:30, 7 September 2024
mediated by alpha-adrenergic receptor activation. Our understanding of the mechanism of drug-induced receptor activation and receptor theory and the biochemical...
33 KB (3,845 words) - 01:47, 19 August 2024
mouth and has a minimal effect on cardiac function due to its α1-adrenergic receptor selectivity. When prazosin is started, however, heart rate and contractility...
21 KB (1,778 words) - 14:23, 29 May 2024