Gabapentin, sold under the brand name Neurontin among others, is an anticonvulsant medication primarily used to treat partial seizures and neuropathic...

gabapentin. It was designed for increased oral bioavailability over gabapentin, and human trials showed it to produce extended release of gabapentin with...

United States in 2004. It was developed as a successor to the related gabapentin. It is available as a generic medication. In 2022, it was the 91st most...

the gabapentin receptor (α2δ subunit), as it is the target of the drugs gabapentin and pregabalin. Clinically used gabapentinoids include gabapentin, pregabalin...

seizures and severe agitation. Approved: Gabapentin (Neurontin) Gabapentin enacarbil (Horizant, Regnite) Gabapentin Extended-Release (Gralise) Pregabalin...

used transdermally (applied topically to the skin) in combination with gabapentin and clonidine prepared at a compounding pharmacy. Common side effects...

Phenibut also binds to and blocks α2δ subunit-containing VDCCs, similarly to gabapentin and pregabalin, and hence is a gabapentinoid. Both (R)-phenibut and (S)-phenibut...

disorder. Curry, W. J; Kulling, D. L (1998). "Newer antiepileptic drugs: Gabapentin, lamotrigine, felbamate, topiramate and fosphenytoin". American Family...

Pregabalin (2004) Mirogabalin (2019) (Japan only) Gabapentin (1993) Gabapentin enacarbil (Horizant) (2011) Gabapentin extended release (Gralise) (1996) Gabapentinoids...

inhibitor and GABA reuptake inhibitor Gabapentin – anticonvulsant; inhibitor of α2δ subunit-containing VGCCs Gabapentin enacarbil – used for the treatment...

to gabapentin, which similarly binds to the α2δ calcium channels (1 and 2). It was developed as a potentially more potent successor to gabapentin and...

4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...

most widely attempted medication is gabapentin, with one case series finding that seven of eight patients on gabapentin showed improvement in attack frequency...

4-Methylpregabalin Arbaclofen Arbaclofen placarbil Atagabalin Baclofen Gabapentin Gabapentin enacarbil Imagabalin Mirogabalin PD-200,347 PD-217,014 PD-299,685...

Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin Antidepressants SSRIsTooltip Selective...

pharmaceutical marketing. In 1993, the Food and Drug Administration (FDA) approved gabapentin only for treatment of seizures. Warner–Lambert, which merged with Pfizer...

short trial period of gabapentin therapy is recommended, to determine the effectiveness for that person. 62% of people taking gabapentin may have at least...

consisting of a combination of hydroxyzine and two other medications (gabapentin and flumazenil) as well as therapy, is an ineffective treatment promoted...

severe allergic reactions due to its strong antihistamine properties. Gabapentin, approved for treatment of seizures and postherpetic neuralgia in adults...

Etifoxine Hypnotics Zopiclone Gabapentinoids (α2δ VDCC blockers) Gabapentin Gabapentin enacarbil Phenibut Pregabalin Antidepressants SSRIsTooltip Selective...

anti-convulsant medications gabapentin and pregabalin may be used to reduce pain. There is tentative evidence that gabapentin may be of benefit for pain...

S2CID 34610971. Matsuda KM, Sharma D, Schonfeld AR, Kwatra SG (September 2016). "Gabapentin and pregabalin for the treatment of chronic pruritus". Journal of the...

with newer anti-seizure medications such as gabapentin, offer a possible regimen for seizure control. Gabapentin has the additional feature of aiding in the...

advantage over certain anxiolytic medications such as benzodiazepines. Gabapentin (Neurontin), a closely related medication to pregabalin with the same...

(duloxetine, venlafaxine, and milnacipran) and antiepileptic medications (gabapentin, pregabalin, oxcarbazepine zonisamide levetiracetam, lamotrigine, topiramate...

hot flashes include cognitive-behavioral therapy, clinical hypnosis, gabapentin, fezolinetant or selective serotonin reuptake inhibitors. These will not...

has been used successfully. Other drugs with variable success include gabapentin and, recently,[when?] memantine. Successful surgery options include superior...

non-steroidal anti-inflammatory drugs (NSAIDs), prostaglandin-based drugs, gabapentin, and methylcobalamin. However, the quality of evidence supporting their...

propanamide does not change after Hofmann reaction. In the synthesis of gabapentin, beginning with the mono-amidation of 1,1-cyclohexane diacetic acid anhydride...

dopamine agonists like pramipexole and gabapentinoids (α2δ ligands) like gabapentin. RLS affects an estimated 2.5–15% of the American population. Females...