A prodrug is a pharmacologically inactive medication or compound that, after intake, is metabolized (i.e., converted within the body) into a pharmacologically...

neurotransmitter prodrug, or neurotransmitter precursor, is a drug that acts as a prodrug of a neurotransmitter. A variety of neurotransmitter prodrugs have been...

Directed enzyme prodrug therapy (DEPT) uses enzymes artificially introduced into the body to convert prodrugs, which have no or poor biologically activity...

of mometasone, is the marketed medication. Mometasone furoate acts as a prodrug of mometasone. In addition to its glucocorticoid activity, mometasone also...

psilocybin for pharmacological studies, as they are both believed to be prodrugs of psilocin. However, some users report that O-acetylpsilocin's subjective...

(γ-hydroxybutyric acid acetate) – synthetic prodrug to GHB GBL (γ-hydroxybutyric acid lactone) – metabolic intermediate and prodrug to GHB GHBAL (γ-hydroxybutyraldehyde...

estrogen in such research. However, NETE, an intramuscularly administered prodrug of norethisterone which is used as a long-acting contraceptive, is used...

Hypoxia-Activated Prodrugs (HAPs) are prodrugs that target regions of tumor hypoxia within tumor cells. HAPs may offer the potential, alone and in combination...

Levomethorphan is a prodrug to levorphanol, analogously to DXM acting as a prodrug to dextrorphan or codeine behaving as a prodrug to morphine. As such...

damage. Boldenone undecylenate is an androgen ester and a long-lasting prodrug of boldenone in the body. Boldenone undecylenate was introduced for medical...

called prodrugs. The reasons for this type of formulation may be because the drug is more stable during manufacture and storage as the prodrug form, or...

This is a list of androgens/anabolic steroids (AAS) or testosterone derivatives. Androgen esters are mostly not included in this list. The major classes...

Corticosteroids are a class of steroid hormones that are produced in the adrenal cortex of vertebrates, as well as the synthetic analogues of these hormones...

N-diisopropyltryptamine) is a psychedelic tryptamine derivative which is a prodrug ester of the well known designer drug 4-HO-DiPT. It is one of a number...

bacterium Moraxella catarrhalis. Tributyrin is a stable and rapidly absorbed prodrug of butyric acid which enhances antiproliferative effects of dihydroxycholecalciferol...

His main research focus has been on the design and characterization of prodrugs and protoxins targeted for activation by cancer specific proteases. This...

modulators mAChRsTooltip Muscarinic acetylcholine receptors Precursors (and prodrugs) Acetyl-coA Adafenoxate Choline (lecithin) Citicoline Cyprodenate Dimethylethanolamine...

the lysine-analog of enalapril. Unlike other ACE inhibitors, it is not a prodrug, is not metabolized by the liver, and is excreted unchanged in the urine...

glucocorticoid effects. Trenbolone acetate is an androgen ester and a short-lasting prodrug of trenbolone in the body. Trenbolone acetate was discovered in 1963 and...

olmesartan, the metabolism of the drug is unusual as it is a cascading prodrug. Candesartan has good bioavailibility and is the most potent by weight...

dipropionate is the USAN and former BAN. It is a prodrug of the free form, beclometasone (INN). The prodrug beclometasone is marketed in Norway and Russia...

an androgen and testosterone prodrug Δ1-Androstenediol (Δ1-androsten-3β,17β-diol) – an androgen and δ1-testosterone prodrug Androstenedione Δ4-Androstenedione...

received regulatory approval in 1991. Nabumetone is a non-acidic NSAID prodrug that is rapidly metabolized in the liver to the active metabolite, 6-methoxy-2-naphthyl...

is not recommended by the manufacturer. Lisdexamfetamine is an inactive prodrug that works after being converted by the body into dextroamphetamine, a...

recreational use. γ-Valerolactone (GVL) acts as a prodrug to GHV, analogously to how γ-butyrolactone (GBL) is a prodrug to GHB. 1,4-Butanediol (1-4-BD) Aceburic...

medicine used to treat (chronic) infections with hepatitis B virus. A prodrug form of adefovir was previously called bis-POM PMEA, with trade names Preveon...

Serdexmethylphenidate is a prodrug of dexmethylphenidate created by the pharmaceutical company KemPharm (now Zevra Therapeutics). The compound was first...

N-Phenylacetyl-l-prolylglycine ethyl ester is promoted as a nootropic and is a prodrug of cyclic glycine-proline. Other names include the brand name Noopept (Russian:...

the European Union in February 1996. It was initially introduced as the prodrug mycophenolate mofetil (MMF, trade name CellCept) to improve oral bioavailability...

been evaluated in the treatment of solid tumors, as a hypoxia-activated prodrug (HAPs), such chemical agents in low oxygen conditions undergo bio-reduction...