The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated...
24 KB (2,820 words) - 05:34, 10 July 2024
prescribed in 1934. Progesterone is the most important progestogen in the body. As a potent agonist of the nuclear progesterone receptor (nPR) (with an affinity...
123 KB (11,583 words) - 02:59, 21 December 2024
Membrane progesterone receptors (mPRs) are a group of cell surface receptors and membrane steroid receptors belonging to the progestin and adipoQ receptor (PAQR)...
22 KB (2,417 words) - 07:41, 27 December 2023
Antiprogestogen (redirect from Progesterone receptor antagonist)
drugs competitively inhibit progestin at progesterone receptors, acting by blocking the progesterone receptor (PR) and/or inhibiting or suppressing progestogen...
5 KB (392 words) - 20:56, 24 November 2024
A selective progesterone receptor modulator (SPRM) is an agent that acts on the progesterone receptor (PR), the biological target of progestogens like...
47 KB (5,150 words) - 21:22, 21 November 2024
or an agonist of the progesterone receptor, the biological target of progestogens like endogenous progesterone. Progesterone also has antimineralocorticoid...
175 KB (18,968 words) - 15:19, 3 July 2024
National Laboratory, whose work in isolating and characterizing the progesterone receptor gene has stimulated advances in breast biology and oncology. She...
20 KB (1,818 words) - 03:47, 5 December 2024
synthetic steroid hormones that bind to and activate the progesterone receptors (PR). Progesterone is the major and most important progestogen in the body...
16 KB (1,567 words) - 01:04, 8 October 2024
hence is an agonist of the progesterone receptor (PR), the biological target of progestogens like endogenous progesterone. It opposes the effects of estrogens...
185 KB (18,508 words) - 13:32, 2 November 2024
The progesterone receptor A (PR-A) is one of three known isoforms of the progesterone receptor (PR), the main biological target of the endogenous progestogen...
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receptor (MR; NR3C2) (Aldosterone) 3: Progesterone receptor (PR; NR3C3, PGR) (Sex hormones: Progesterone) 4: Androgen receptor (AR; NR3C4, AR) (Sex hormones:...
23 KB (2,796 words) - 19:08, 19 February 2024
17α-Hydroxyprogesterone (redirect from 17-OH-progesterone)
progesterone receptor (PR) similarly to progesterone, albeit weakly in comparison. In addition, it is an antagonist of the mineralocorticoid receptor...
14 KB (1,126 words) - 10:08, 7 July 2024
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. The medication is an atypical progestogen...
61 KB (6,712 words) - 07:01, 27 October 2024
The progesterone receptor C (PR-C) is one of three known isoforms of the progesterone receptor (PR), the main biological target of the endogenous progestogen...
1 KB (120 words) - 20:17, 13 October 2022
Allopregnanolone (category GABAA receptor positive allosteric modulators)
kainate, and glycine receptors. Unlike progesterone, allopregnanolone is inactive at the classical nuclear progesterone receptor (PR). However, allopregnanolone...
50 KB (4,785 words) - 03:36, 8 December 2024
Mifepristone (category Selective progesterone receptor modulators)
receptor level. In the presence of progesterone, mifepristone acts as a competitive progesterone receptor antagonist (in the absence of progesterone,...
125 KB (11,582 words) - 04:18, 21 December 2024
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has weak androgenic and estrogenic...
95 KB (9,422 words) - 21:09, 24 October 2024
– oral progesterone receptor agonist (progestogen/progestin) for prevention of preterm labor VOLT-02 – water-soluble conjugate of progesterone and neurosteroid...
15 KB (1,238 words) - 22:37, 30 October 2024
Medroxyprogesterone (redirect from Medroxy-progesterone)
(September 2006). "Determination of conformational changes in the progesterone receptor using ELISA-like assays". Steroids. 71 (9): 792–8. doi:10.1016/j...
7 KB (482 words) - 04:13, 23 October 2024
The progesterone receptor B (PR-B) is one of three known isoforms of the progesterone receptor (PR), the main biological target of the endogenous progestogen...
1 KB (120 words) - 20:17, 13 October 2022
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It is a unique progestogen, with strong...
61 KB (5,612 words) - 07:18, 6 November 2024
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has very weak androgenic and glucocorticoid...
63 KB (5,557 words) - 20:17, 5 December 2024
potent progestogenic activity (it binds with high affinity to the progesterone receptor), gynecomastia, characterized by development and swelling of breast...
34 KB (3,265 words) - 04:17, 1 December 2024
Sex-hormonal agent (redirect from Sex-hormone receptor modulator)
hormone receptors. The sex hormones include androgens such as testosterone, estrogens such as estradiol, and progestogens such as progesterone. Sex-hormonal...
5 KB (357 words) - 23:19, 9 May 2024
mediated via the progesterone receptor membrane component-1 (PGRMC1). Certain other progestins act similarly in this assay, whereas progesterone acts neutrally...
83 KB (7,903 words) - 02:07, 10 December 2024
among the highest known affinity of any AAS for the androgen (and progesterone) receptors, and has been said to be perhaps the most potent AAS to have ever...
9 KB (511 words) - 15:49, 24 December 2023
to estrogen receptor positive tumors (i.e. tumors that contain estrogen receptor positive cells), but can also include progesterone receptor positive tumors...
5 KB (508 words) - 10:02, 27 December 2023
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. Due to its androgenic and progestogenic...
21 KB (1,843 words) - 05:55, 16 August 2024
nuclear receptors include members of subfamily 3, such as the androgen receptor, estrogen receptors, glucocorticoid receptor, and progesterone receptor. It...
74 KB (6,689 words) - 16:59, 8 December 2024
Hydroxyprogesterone caproate (redirect from 17-alpha-Hydroxy-progesterone caproate)
progestogen, and hence is an agonist of the progesterone receptor, the biological target of progestogens like progesterone. It has some antimineralocorticoid activity...
121 KB (12,026 words) - 08:48, 2 November 2024