The alpha-2C adrenergic receptor (α2C adrenoceptor), also known as ADRA2C, is an alpha-2 adrenergic receptor, and also denotes the human gene encoding...
13 KB (1,541 words) - 00:52, 27 September 2024
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the human gene encoding it....
12 KB (1,303 words) - 04:16, 13 August 2024
The alpha-2B adrenergic receptor (α2B adrenoceptor), is a G-protein coupled receptor. It is a subtype of the adrenergic receptor family. The human gene...
15 KB (1,754 words) - 20:51, 13 August 2023
The alpha-1D adrenergic receptor (α1D adrenoreceptor), also known as ADRA1D, is an alpha-1 adrenergic receptor, and also denotes the human gene encoding...
10 KB (1,214 words) - 08:14, 12 October 2024
Tizanidine (category Alpha-2 adrenergic receptor agonists)
Tizanidine, sold under the brand name Zanaflex among others, is an alpha-2 (α2) adrenergic receptor agonist, similar to clonidine, that is used to treat muscle...
13 KB (976 words) - 21:26, 28 September 2024
2C or II-C may refer to: 2C (psychedelics), a family of psychedelic phenethylamines Alpha-2C adrenergic receptor in biochemistry Apple IIc, a personal...
975 bytes (167 words) - 10:57, 21 September 2019
Oxymetazoline (category Alpha-1 adrenergic receptor agonists)
adrenergic receptors and α2 adrenergic receptors, most notably. One study classified it in the following order: α(2A) > α(1A) ≥ α(2B) > α(1D) ≥ α(2C)...
14 KB (1,266 words) - 13:55, 14 October 2024
BOH-2C-B, β-Hydroxy-2C-B, βOH-2CB BMB 2C-B-5-hemifly 2C-B-aminorex (2C-B-AR) 2C-B-AN 2C-B-BZP 2C-B-FLY-NB2EtO5Cl 2C-B-PP 2CB-Ind βk-2C-B (beta-keto 2C-B)...
38 KB (4,198 words) - 06:35, 6 October 2024
Guanfacine (category Alpha-2 adrenergic receptor agonists)
(December 1994). "The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors". The Journal...
43 KB (3,962 words) - 17:44, 30 September 2024
Sympathomimetic drug (redirect from Adrenergic agent)
have greater beta adrenergic receptor activity, but if the substituent is not bulky, then it will favor the alpha adrenergic receptors. Direct stimulation...
9 KB (891 words) - 19:06, 3 September 2024
scientists found how evolution has favored low levels of the alpha-2C adrenergic receptor. This protein coding gene helps inhibit the sympathetic nervous...
110 KB (14,485 words) - 21:34, 16 October 2024
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). The 5-HT2A...
90 KB (9,886 words) - 06:08, 13 September 2024
BOH-2C-B, β-Hydroxy-2C-B, βOH-2CB BMB 2C-B-5-hemifly 2C-B-aminorex (2C-B-AR) 2C-B-AN 2C-B-BZP 2C-B-FLY-NB2EtO5Cl 2C-B-PP 2CB-Ind βk-2C-B (beta-keto 2C-B)...
13 KB (1,469 words) - 18:15, 12 September 2024
found that lessen the risk of neurotoxicity from NMDA receptor antagonists. Centrally acting alpha 2 agonists such as clonidine and guanfacine are thought...
38 KB (4,196 words) - 12:46, 14 July 2024
Atipamezole (category Alpha-2 blockers)
sold under the brand name Antisedan among others, is a synthetic α2 adrenergic receptor antagonist used for the reversal of the sedative and analgesic effects...
24 KB (2,110 words) - 00:27, 13 September 2024
to be an active Alpha-1 adrenergic receptor agonist in rabbit ear arteries. It has binding affinity towards 5-HT2C and 5-HT2A receptors in rats. It features...
5 KB (391 words) - 01:06, 21 July 2023
receptors D1 and D2, histamine receptor H1, and A1 adrenoreceptors. Ketanserin Antihypertensive. Blocks 5-HT2A, 5-HT2C and Alpha 1 (A1) adrenoreceptors. Risperidone...
5 KB (503 words) - 03:53, 9 October 2024
also shown to be a partial agonist of adrenergic receptors. A potential risk of neurotoxicity from 2C-T-2 use (and 2C chemical series in general) has been...
12 KB (1,152 words) - 07:24, 16 November 2023
βk-2C-B (βeta-keto-4-bromo-2,5-dimethoxyphenylamine), also known as bk-2C-B, is a novel psychedelic substance. It is the beta (β) ketone structural analogue...
22 KB (2,930 words) - 09:13, 20 October 2024
Lofexidine (category Alpha-2 adrenergic receptor agonists)
is an agonist at the alpha-2A, 2B, and 2C adrenergic receptor subtypes, with the highest activity at the α2A-adrengergic receptor. Ki represents the dissociation...
15 KB (1,396 words) - 22:26, 15 October 2024
Cannabigerol (category Alpha-2 adrenergic receptor agonists)
cannabinoid receptors, where it acts as a weak partial agonist. Conversely, it is a much more potent agonist of the α2-adrenergic receptor, antagonist...
24 KB (1,932 words) - 19:17, 22 September 2024
Phenylephrine (category Alpha-1 adrenergic receptor agonists)
is safe. Phenylephrine is a selective α1-adrenergic receptor agonist with minimal to no β-adrenergic receptor agonist activity or induction of norepinephrine...
57 KB (4,906 words) - 10:33, 4 October 2024
optimum receptor binding at 5-HT2A, but it is still considerably less potent than its alpha-methyl derivative Bromo-DragonFLY. 2C-B-aminorex 2C-B-BUTTERFLY...
3 KB (209 words) - 07:28, 14 February 2024
Mirtazapine (category Alpha-2 blockers)
it works is not clear, but it may involve blocking certain adrenergic and serotonin receptors. Chemically, it is a tetracyclic antidepressant, and is closely...
88 KB (7,952 words) - 16:30, 19 October 2024
2C (2C-x) is a general name for the family of psychedelic phenethylamines containing methoxy groups on the 2 and 5 positions of a benzene ring. Most of...
12 KB (497 words) - 05:26, 21 October 2024
Tyramine (redirect from Tyramine receptor)
secreted into the synapse, and octopamine does not activate alpha or beta adrenergic receptors.[medical citation needed] When using a MAO inhibitor (MAOI)...
28 KB (2,685 words) - 05:20, 28 August 2024
Corbadrine (redirect from Alpha-methylnorepineprine)
agonist of the α1-, α2-, and β-adrenergic receptors. It is said to have preferential activity at the α2-adrenergic receptor. Corbadrine is also a metabolite...
7 KB (423 words) - 05:02, 2 September 2024
various nuclear receptors. The structure of the LBD is referred to as an alpha helical sandwich fold in which three anti parallel alpha helices (the "sandwich...
74 KB (6,683 words) - 09:55, 12 September 2024
Octopamine (redirect from Octopamine receptor β)
into distinct types: OctαR (alpha-adrenergic-like), are structurally and functionally similar to noradrenergic alpha-1 receptors in mammals. There are multiple...
39 KB (4,008 words) - 23:56, 31 August 2024
Methoxamine (category Alpha-1 adrenergic receptor agonists)
It has mostly or entirely been discontinued. The drug is an α1-adrenergic receptor agonist.[additional citation(s) needed] The long duration of action...
8 KB (510 words) - 01:05, 2 September 2024