The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...
25 KB (2,231 words) - 08:33, 22 August 2024
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the human gene encoding it....
12 KB (1,303 words) - 04:16, 13 August 2024
The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline)...
33 KB (2,982 words) - 11:42, 7 August 2024
The alpha-2C adrenergic receptor (α2C adrenoceptor), also known as ADRA2C, is an alpha-2 adrenergic receptor, and also denotes the human gene encoding...
13 KB (1,540 words) - 04:17, 8 March 2024
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are...
16 KB (1,528 words) - 10:28, 23 June 2024
The alpha-2B adrenergic receptor (α2B adrenoceptor), is a G-protein coupled receptor. It is a subtype of the adrenergic receptor family. The human gene...
15 KB (1,754 words) - 20:51, 13 August 2023
The alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic receptor, is an alpha-1 adrenergic...
11 KB (1,360 words) - 10:20, 23 June 2024
Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor...
13 KB (1,364 words) - 03:02, 21 August 2024
Antihypertensive (redirect from Alpha-2 adrenergic receptor agonist)
beta-2-adrenergic receptors reduce blood pressure through increased relaxation of smooth muscle. Alpha-blockers can block alpha-1 adrenergic receptors and/or...
56 KB (6,323 words) - 16:42, 23 August 2024
The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...
33 KB (3,380 words) - 19:17, 10 July 2024
adrenergic receptor (β1 adrenoceptor), also known as ADRB1, can refer to either the protein-encoding gene (gene ADRB1) or one of the four adrenergic receptors...
31 KB (3,743 words) - 00:48, 23 July 2024
The alpha-1B adrenergic receptor (α1B-adrenoreceptor), also known as ADRA1B, is an alpha-1 adrenergic receptor, and also denotes the human gene encoding...
11 KB (1,333 words) - 02:33, 18 October 2022
receptor. Beta-3 adrenergic receptor has been shown to interact with Src. Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor...
17 KB (2,039 words) - 09:45, 7 October 2023
pharmacological agents that act as antagonists on α-adrenergic receptors (α-adrenoceptors). Historically, alpha-blockers were used as a tool for pharmacologic...
34 KB (3,210 words) - 22:18, 7 August 2024
The alpha-1D adrenergic receptor (α1D adrenoreceptor), also known as ADRA1D, is an alpha-1 adrenergic receptor, and also denotes the human gene encoding...
8 KB (1,043 words) - 04:13, 8 March 2024
Methyldopa (redirect from Alpha-methyldopa)
liver problems, and allergic reactions. Methyldopa is in the alpha-2 adrenergic receptor agonist family of medication. It works by stimulating the brain...
13 KB (1,020 words) - 08:17, 12 June 2024
first group of receptors are the beta (β) adrenergic receptors. There are β1, β2, and β3 receptors. The second group contains the alpha (α) adrenoreceptors...
15 KB (1,535 words) - 19:07, 2 August 2024
Alpha-2 blockers (or α2 blockers) are a subset of the alpha blocker class of drugs and are antagonists to the α2 adrenergic receptor. They are mainly used...
3 KB (339 words) - 18:58, 20 August 2024
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of adrenergic receptors are: α1, α2...
7 KB (750 words) - 04:55, 1 April 2024
Guanfacine (category Alpha-2 adrenergic receptor agonists)
pregnancy or breastfeeding. It appears to work by activating α2A-adrenergic receptors in the brain, thereby decreasing sympathetic nervous system activity...
43 KB (3,962 words) - 20:10, 8 August 2024
Tizanidine (category Alpha-2 adrenergic receptor agonists)
Tizanidine, sold under the brand name Zanaflex among others, is an alpha-2 (α2) adrenergic receptor agonist, similar to clonidine, that is used to treat muscle...
13 KB (972 words) - 16:25, 28 June 2024
stress disorder. Alpha-1 adrenergic receptors are present in vascular smooth muscle, the central nervous system, and other tissues. When alpha blockers bind...
38 KB (4,243 words) - 20:56, 27 November 2023
Adrenergic means "working on adrenaline (epinephrine) or noradrenaline (norepinephrine)" (or on their receptors). When not further qualified, it is usually...
3 KB (284 words) - 18:10, 25 July 2024
fiction anthology edited by Robert Silverberg Alpha-2 adrenergic receptor, a protein family ISO 3166-1 alpha-2, two-letter country codes as assigned by the International...
368 bytes (80 words) - 19:40, 8 April 2024
Clonidine (redirect from Catapres-tts-2)
PMID 9374795. Giovannitti JA, Thoms SM, Crawford JJ (2015). "Alpha-2 adrenergic receptor agonists: a review of current clinical applications". Anesthesia...
60 KB (5,506 words) - 21:49, 10 July 2024
Beta blocker (redirect from Beta-adrenergic receptor antagonists)
and β3 receptors.: 153 β1-adrenergic receptors are located mainly in the heart and in the kidneys. β2-adrenergic receptors are located mainly in the lungs...
75 KB (7,456 words) - 02:29, 6 August 2024
Xylometazoline (category Alpha-2 adrenergic receptor agonists)
decongestant and alpha-adrenergic agonist families of medication. One study classified it with selectivity ratios in alpha 2 adrenergic receptors of 151 for...
14 KB (1,107 words) - 13:34, 21 August 2024
Oxymetazoline (category Alpha-2 adrenergic receptor agonists)
classified it with selectivity ratios in alpha 2 adrenergic receptors of 200 for a2A vs a2B, 7.1 a2A vs a2C, and 28.2 a2B vs a2C. In 2021, it was the 292nd...
15 KB (1,266 words) - 05:55, 14 May 2024
Amitraz (category Alpha-2 adrenergic receptor agonists)
synergist. Its effectiveness is traced back on alpha-adrenergic agonist activity, interaction with octopamine receptors of the central nervous system and inhibition...
31 KB (3,737 words) - 18:35, 15 July 2024
Xylazine (category Alpha-2 adrenergic receptor agonists)
Xylazine is a structural analog of clonidine and an alpha-2 adrenergic receptor agonist, sold under many trade names worldwide, most notably the Bayer...
42 KB (4,337 words) - 07:49, 21 August 2024