Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has...
13 KB (1,364 words) - 06:38, 1 April 2024
The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...
25 KB (2,231 words) - 23:55, 13 July 2024
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of adrenergic receptors are: α1, α2...
7 KB (750 words) - 04:55, 1 April 2024
Beta adrenergic agonists or beta agonists are medications that relax muscles of the airways, causing widening of the airways and resulting in easier breathing...
9 KB (805 words) - 20:40, 27 May 2024
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are...
16 KB (1,528 words) - 10:28, 23 June 2024
Alpha agonist may refer to: Alpha-adrenergic agonist, drugs that selectively stimulate alpha adrenergic receptors PPAR-alpha agonist, drugs which act upon...
246 bytes (60 words) - 06:54, 14 August 2020
Xylometazoline (category Alpha-1 adrenergic receptor agonists)
decongestant and alpha-adrenergic agonist families of medication. One study classified it with selectivity ratios in alpha 2 adrenergic receptors of 151...
13 KB (1,079 words) - 12:12, 6 August 2024
Metaraminol (category Alpha-1 adrenergic receptor agonists)
have direct alpha-adrenergic agonist and β1 adrenergic agonist effects. However at doses common in clinical practice, the indirect α1 adrenergic effects predominate...
8 KB (491 words) - 20:50, 22 October 2023
β1-Adrenergic receptor agonists, also known as beta-1 agonists, are a class of drugs that bind selectively to the β1-adrenergic receptor. As a result,...
4 KB (322 words) - 00:48, 23 July 2024
selective alpha-1 antagonists are available. As of 2018, prazosin is the only alpha-1 blocker known to act as an inverse agonist at all alpha-1 adrenergic receptor...
38 KB (4,243 words) - 20:56, 27 November 2023
but also many medications like beta blockers, beta-2 (β2) agonists and alpha-2 (α2) agonists, which are used to treat high blood pressure and asthma, for...
33 KB (2,982 words) - 11:42, 7 August 2024
The alpha-1A adrenergic receptor (α1A adrenoreceptor), also known as ADRA1A, formerly known also as the alpha-1C adrenergic receptor, is an alpha-1 adrenergic...
11 KB (1,360 words) - 10:20, 23 June 2024
(antidepressant) Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-2 adrenergic receptor Beta-3 adrenergic receptor GRCh38:...
31 KB (3,743 words) - 00:48, 23 July 2024
PMID 18092107. Giovannitti JA, Thoms SM, Crawford JJ (2015). "Alpha-2 adrenergic receptor agonists: a review of current clinical applications". Anesth Prog...
15 KB (1,535 words) - 19:07, 2 August 2024
Tizanidine (category Alpha-2 adrenergic receptor agonists)
sold under the brand name Zanaflex among others, is an alpha-2 (α2) adrenergic receptor agonist, similar to clonidine, that is used to treat muscle spasticity...
13 KB (972 words) - 16:25, 28 June 2024
Amitraz (category Alpha-2 adrenergic receptor agonists)
as a pesticide synergist. Its effectiveness is traced back on alpha-adrenergic agonist activity, interaction with octopamine receptors of the central...
31 KB (3,737 words) - 18:35, 15 July 2024
Beta blocker (redirect from Beta-adrenergic blocker)
Beta blockers must not be used in the treatment of selective alpha-adrenergic agonist overdose. The blockade of only beta receptors increases blood pressure...
75 KB (7,456 words) - 02:29, 6 August 2024
α1B-adrenergic receptor has been determined in complex with the inverse agonist (+)-cyclazosin. There are 3 alpha-1 adrenergic receptor subtypes: alpha-1A...
11 KB (1,333 words) - 02:33, 18 October 2022
The alpha-2C adrenergic receptor (α2C adrenoceptor), also known as ADRA2C, is an alpha-2 adrenergic receptor, and also denotes the human gene encoding...
13 KB (1,540 words) - 04:17, 8 March 2024
Sympathomimetic drug (redirect from Adrenergic agent)
drugs (also known as adrenergic drugs and adrenergic amines) are stimulant compounds which mimic the effects of endogenous agonists of the sympathetic nervous...
9 KB (891 words) - 12:49, 14 July 2024
Norepinephrine (category Alpha-adrenergic agonists)
norepinephrine receptors have been identified, known as alpha and beta adrenergic receptors. Alpha receptors are divided into subtypes α1 and α2; beta receptors...
59 KB (6,525 words) - 20:54, 14 August 2024
Antihypertensive drug (redirect from Alpha-2 adrenergic receptor agonist)
PMID 12748199. Giovannitti JA, Thoms SM, Crawford JJ (2015). "Alpha-2 adrenergic receptor agonists: a review of current clinical applications". Anesthesia Progress...
56 KB (6,323 words) - 13:32, 11 August 2024
Adrenaline (category Alpha-adrenergic agonists)
muscle that lines most arterioles. Adrenaline is a nonselective agonist of all adrenergic receptors, including the major subtypes α1, α2, β1, β2, and β3...
57 KB (6,552 words) - 19:02, 9 August 2024
receptor. Beta-3 adrenergic receptor has been shown to interact with Src. Other adrenergic receptors Alpha-1 adrenergic receptor Alpha-2 adrenergic receptor Beta-1...
17 KB (2,039 words) - 09:45, 7 October 2023
adrenergic receptor Alpha-2 adrenergic receptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor Discovery and development of beta2 agonists GRCh38: Ensembl...
33 KB (3,380 words) - 19:17, 10 July 2024
Sympatholytic (redirect from Adrenergic neurone blockers)
cellular signaling pathways of adrenergic receptors. However, there are exceptions: clonidine is an adrenergic agonist at the α2 receptor; since this...
11 KB (1,303 words) - 21:40, 3 December 2023
Guanfacine (category Alpha-2 adrenergic receptor agonists)
(immediate-release) and Intuniv (extended-release) among others, is an oral alpha-2a agonist medication used to treat attention deficit hyperactivity disorder (ADHD)...
43 KB (3,962 words) - 20:10, 8 August 2024
Prazosin (category Alpha-1 blockers)
control nasal vascular blood flow and alpha blockers inhibit this, in the same way that alpha-adrenergic agonists have the opposite effect of being a decongestant...
21 KB (1,778 words) - 14:23, 29 May 2024
The alpha-2B adrenergic receptor (α2B adrenoceptor), is a G-protein coupled receptor. It is a subtype of the adrenergic receptor family. The human gene...
15 KB (1,754 words) - 20:51, 13 August 2023
Isoprenaline (category Alpha-adrenergic agonists)
others. Isoprenaline is a selective agonist of the β-adrenergic receptors, including both the β1- and β2-adrenergic receptors. By activating these receptors...
33 KB (2,785 words) - 06:06, 12 August 2024