The beta-2 adrenergic receptor (β2 adrenoreceptor), also known as ADRB2, is a cell membrane-spanning beta-adrenergic receptor that binds epinephrine (adrenaline)...
33 KB (3,380 words) - 19:17, 10 July 2024
The beta-3 adrenergic receptor (β3-adrenoceptor), also known as ADRB3, is a beta-adrenergic receptor, and also denotes the human gene encoding it. Actions...
17 KB (2,039 words) - 09:45, 7 October 2023
The beta-1 adrenergic receptor (β1 adrenoceptor), also known as ADRB1, can refer to either the protein-encoding gene (gene ADRB1) or one of the four adrenergic...
31 KB (3,743 words) - 00:48, 23 July 2024
Beta adrenergic agonists or beta agonists are medications that relax muscles of the airways, causing widening of the airways and resulting in easier breathing...
9 KB (805 words) - 20:40, 27 May 2024
The alpha-2 (α2) adrenergic receptor (or adrenoceptor) is a G protein-coupled receptor (GPCR) associated with the Gi heterotrimeric G-protein. It consists...
25 KB (2,231 words) - 23:55, 13 July 2024
The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline)...
33 KB (2,982 words) - 15:38, 5 June 2024
A Beta-2 adrenergic antagonist (β2-adrenoceptor antagonist) is an adrenergic antagonist which blocks the beta-2 adrenergic receptors of cells, with either...
1 KB (104 words) - 20:58, 12 August 2023
types of β-adrenergic receptors and others are selective for one of the three known types of beta receptors, designated β1, β2 and β3 receptors.: 153 β1-adrenergic...
72 KB (7,108 words) - 07:21, 15 July 2024
Beta2-adrenergic agonists, also known as adrenergic β2 receptor agonists, are a class of drugs that act on the β2 adrenergic receptor. Like other β adrenergic...
18 KB (1,703 words) - 06:18, 17 March 2024
into two groups. The first group of receptors are the beta (β) adrenergic receptors. There are β1, β2, and β3 receptors. The second group contains the alpha...
14 KB (1,465 words) - 22:49, 25 June 2024
alpha-1 (α1) adrenergic receptors are G protein-coupled receptors (GPCRs) associated with the Gq heterotrimeric G protein. α1-adrenergic receptors are subdivided...
16 KB (1,528 words) - 10:28, 23 June 2024
2000). "The interaction of beta-arrestin with the AP-2 adaptor is required for the clustering of beta 2-adrenergic receptor into clathrin-coated pits"...
82 KB (9,384 words) - 18:56, 11 June 2024
The alpha-2A adrenergic receptor (α2A adrenoceptor), also known as ADRA2A, is an α2 adrenergic receptor, and also denotes the human gene encoding it. α2...
12 KB (1,307 words) - 05:44, 17 May 2024
G-protein-coupled receptor kinase 2 (GRK2) is an enzyme that in humans is encoded by the ADRBK1 gene. GRK2 was initially called Beta-adrenergic receptor kinase (βARK...
14 KB (1,637 words) - 11:17, 19 June 2022
Alpha-adrenergic agonists are a class of sympathomimetic agents that selectively stimulates alpha adrenergic receptors. The alpha-adrenergic receptor has...
13 KB (1,364 words) - 06:38, 1 April 2024
signalling roles in their own right. Arrestin beta 2, like arrestin beta 1, was shown to inhibit beta-adrenergic receptor function in vitro. It is expressed at...
17 KB (1,962 words) - 03:34, 6 May 2024
G-protein-coupled receptor kinase 3 (GRK3) is an enzyme that in humans is encoded by the ADRBK2 gene. GRK3 was initially called Beta-adrenergic receptor kinase 2 (βARK-2)...
16 KB (2,012 words) - 14:01, 20 January 2024
Beta 2 (β2), may stand for: Beta-2 adrenergic receptor Beta 2 Limited NeuroD1, transcription factor TGF beta 2 This disambiguation page lists articles...
365 bytes (51 words) - 18:18, 18 July 2022
Antihypertensive drug (redirect from Alpha-2 adrenergic receptor agonist)
disease. Beta-blockers can block beta-1 adrenergic receptors and/or beta-2 adrenergic receptors. Those that block beta-1-adrenergic receptors prevent the...
56 KB (6,323 words) - 15:08, 21 July 2024
and acts as a cofactor in the beta-adrenergic receptor kinase (BARK) mediated desensitization of beta-adrenergic receptors. Besides the central nervous...
14 KB (1,584 words) - 01:36, 29 May 2023
An adrenergic agonist is a drug that stimulates a response from the adrenergic receptors. The five main categories of adrenergic receptors are: α1, α2...
7 KB (750 words) - 04:55, 1 April 2024
enzymology, a beta-adrenergic-receptor kinase (EC 2.7.11.15) is an enzyme that catalyzes the chemical reaction: ATP + [beta-adrenergic receptor] ⇌ {\displaystyle...
4 KB (381 words) - 13:18, 26 August 2023
Adrenergic receptor autoantibodies The adrenergic receptors (or adrenoreceptors) are a class of cell membrane-bound protein receptors throughout the body...
15 KB (1,636 words) - 05:57, 15 April 2024
Tachyphylaxis (section Beta-2 agonists)
beta-2 adrenergic receptor, such as salbutamol (albuterol in the US), is the most common treatment for asthma. Polymorphisms of the beta-2 receptor play...
13 KB (1,372 words) - 01:50, 29 April 2024
Bisoprolol (category Beta blockers)
under the brand name Zebeta among others, is a beta blocker which is selective for the beta-1 receptor and used for cardiovascular diseases, including...
31 KB (2,865 words) - 06:05, 26 July 2024
The β3 (beta 3) adrenergic receptor agonist or β3-adrenoceptor agonist, also known as β3-AR agonist, are a class of medicine that bind selectively to...
21 KB (2,188 words) - 03:36, 20 October 2023
Sympatholytic (redirect from Adrenergic neurone blockers)
norepinephrine. They are primarily postsynaptic adrenergic receptor antagonists (alpha and beta adrenergic receptor antagonists, or "blockers"), inhibiting the...
11 KB (1,303 words) - 21:40, 3 December 2023
specific types of adrenergic blockers used, including alpha 1, alpha 2, beta 1, and beta 2. There are various labeled uses of adrenergic neurone blockers...
18 KB (1,925 words) - 05:54, 29 November 2023
Sympathomimetic drug (redirect from Adrenergic agent)
have greater beta adrenergic receptor activity, but if the substituent is not bulky, then it will favor the alpha adrenergic receptors. Direct stimulation...
9 KB (891 words) - 12:49, 14 July 2024
β adrenergic receptor antagonists (also called beta-blockers or β-blockers) were initially developed in the 1960s, for the treatment of angina pectoris...
36 KB (4,063 words) - 07:02, 11 December 2023