= 98% E-6837 – Full agonist at human 5HT6 receptors E-6801 E-6837 – partial agonist at rat 5-HT6 receptors. Orally active in rats, and caused weight loss...
29 KB (3,308 words) - 15:33, 22 September 2024
which activates 5-HT1A, 5-HT1D, 5-HT1B, D2 and norepinephrine receptors. LSD (a psychedelic) is a 5-HT1A, 5-HT2A, 5-HT2C, 5-HT5A and 5-HT6 agonist. The genes...
65 KB (5,263 words) - 07:14, 24 November 2024
5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
2 KB (166 words) - 00:47, 13 May 2022
of 5-HT3 receptors in cell lines and native tissues quickly followed. 5-HT1 receptor 5-HT2 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7...
22 KB (2,395 words) - 18:29, 18 July 2024
articles of the individual subtypes: 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Hoyer D, Clarke DE, Fozard JR...
5 KB (472 words) - 12:54, 25 December 2023
Paliperidone Risperidone 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor GRCh38: Ensembl release...
25 KB (2,992 words) - 06:56, 16 November 2024
Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
18 KB (2,074 words) - 04:01, 28 October 2024
206 nM affinity. SB-699,551 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
15 KB (1,674 words) - 17:31, 10 November 2024
a 5-HT5A receptor agonist, and this action could be involved in the sleep-promoting effects of valerian. No selective agonists of the 5-HT6 receptor have...
16 KB (1,669 words) - 22:38, 28 November 2024
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). The 5-HT2A...
91 KB (9,998 words) - 02:02, 29 November 2024
The 5-HT2C receptor is a subtype of the 5-HT2 receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). Like all 5-HT2...
51 KB (6,108 words) - 22:22, 24 November 2024
receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter. 5-HT1A...
58 KB (6,188 words) - 15:33, 22 September 2024
The 5-HT3 antagonists, informally known as "setrons", are a class of drugs that act as receptor antagonists at the 5-HT3 receptor, a subtype of serotonin...
43 KB (4,628 words) - 19:53, 18 December 2024
5-Benzyloxytryptamine (5-BT), is a tryptamine derivative which acts as an agonist at the 5-HT1D, 5-HT2 and 5-HT6 serotonin receptors, and an antagonist...
4 KB (255 words) - 17:22, 12 June 2024
5-hydroxytryptamine receptor 1B also known as the 5-HT1B receptor is a protein that in humans is encoded by the HTR1B gene. The 5-HT1B receptor is a 5-HT...
22 KB (2,445 words) - 05:54, 16 December 2024
5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT2B is a member...
79 KB (7,607 words) - 21:37, 30 November 2024
5-HT2C receptor agonists are a class of drugs that activate 5-HT2C receptors. They have been investigated for the treatment of a number of conditions including...
48 KB (5,032 words) - 18:40, 8 March 2024
Gs alpha subunit (section Receptors)
protein-coupled receptors that couple to the Gs family proteins include: 5-HT4, 5-HT6 and 5-HT7 serotonergic receptors Adenosine receptor types A2a and...
6 KB (719 words) - 12:10, 31 July 2024
EMDT (redirect from 2-Ethyl-5-methoxy-N,N-dimethyltryptamine)
2-Ethyl-5-methoxy-N,N-dimethyltryptamine (EMDT) is a tryptamine derivative which is used in scientific research. It acts as a selective 5-HT6 receptor agonist...
3 KB (239 words) - 05:50, 1 June 2023
5-hydroxytryptamine (serotonin) receptor 1F, also known as HTR1F is a 5-HT1 receptor protein and also denotes the human gene encoding it. 5-n-Butyryloxy-DMT:...
9 KB (1,053 words) - 15:17, 26 November 2023
Hypidone (category 5-HT6 agonists)
disorder. It acts as a serotonin reuptake inhibitor, 5-HT1A receptor partial agonist, and 5-HT6 receptor full agonist. It is used as the hydrochloride salt...
6 KB (306 words) - 20:52, 5 April 2024
SB-399885 (category 5-HT6 antagonists)
a potent, selective and orally active 5-HT6 receptor antagonist, with a Ki of 9.0nM. SB-399885 and other 5-HT6 antagonists show nootropic effects in animal...
5 KB (365 words) - 15:59, 23 September 2024
5-hydroxytryptamine (serotonin) receptor 1D, also known as HTR1D, is a 5-HT receptor, but also denotes the human gene encoding it. 5-HT1D acts on the central...
11 KB (1,238 words) - 09:14, 27 October 2024
SB-258585 (category 5-HT6 antagonists)
orally active 5-HT6 receptor antagonist, with a Ki of 8.9nM. It is used in its 125I radiolabelled form to map the distribution of 5-HT6 receptors in the brain...
5 KB (393 words) - 15:57, 23 September 2024
the treatment of agitation in Alzheimer's dementia. It is a selective 5-HT6 receptor antagonist. "Masupirdine - Suven Life Sciences". AdisInsight. Springer...
2 KB (80 words) - 12:07, 25 October 2024
PRX-07034 is a selective 5-HT6 receptor antagonist. It has cognition and memory-enhancing properties and potently decreases food intake and body weight...
5 KB (273 words) - 09:25, 16 October 2022
E-6801 (category 5-HT6 agonists)
E-6801 is a partial agonist of the 5-HT6 receptor. It enhanced recognition memory and reversed the memory deficits of scopolamine in an object recognition...
2 KB (130 words) - 09:52, 25 May 2023
EMD-386088 (category 5-HT6 agonists)
research. It acts as a potent 5-HT6 receptor partial agonist, with a Ki of 1 nM, a significantly higher affinity than older 5-HT6 agonists such as EMDT, although...
3 KB (218 words) - 19:01, 25 September 2024
Ro 04-6790 (category 5-HT6 antagonists)
potent and selective receptor antagonist for the 5-HT6 serotonin receptor subtype, with little or no affinity at other receptors. In common with other...
3 KB (264 words) - 19:41, 20 December 2023
μ, δ1, δ2, κ Serotonergic: 5-HT1A, 5-HT1B, 5-HT1D, 5-HT1E, 5-HT1F, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT3, 5-HT4, 5-HT5, 5-HT6, 5-HT7 Autoreceptor Catecholamines...
16 KB (1,590 words) - 01:49, 26 October 2023