The 5-HT7 receptor is a member of the GPCR superfamily of cell surface receptors and is activated by the neurotransmitter serotonin (5-hydroxytryptamine...
25 KB (2,990 words) - 04:12, 19 February 2024
5-HT2A receptor 5-HT2B receptor 5-HT2C receptor 5-HT1 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Category:5-HT2...
2 KB (166 words) - 00:47, 13 May 2022
The 5-HT2A receptor is a subtype of the 5-HT2 receptor that belongs to the serotonin receptor family and is a G protein-coupled receptor (GPCR). The 5-HT2A...
87 KB (9,542 words) - 04:09, 8 August 2024
articles of the individual subtypes: 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor Hoyer D, Clarke DE, Fozard JR...
5 KB (472 words) - 12:54, 25 December 2023
5-HT3 receptors in cell lines and native tissues quickly followed. 5-HT1 receptor 5-HT2 receptor 5-HT4 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor...
22 KB (2,395 words) - 18:29, 18 July 2024
206 nM affinity. SB-699,551 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT4 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
15 KB (1,666 words) - 15:17, 26 November 2023
receptor (or 5-HT1A receptor) is a subtype of serotonin receptors, or 5-HT receptors, that binds serotonin, also known as 5-HT, a neurotransmitter. 5-HT1A...
58 KB (6,181 words) - 22:24, 4 August 2024
Chamomile (ethanol extract) 5-HT receptor 5-HT1 receptor 5-HT2 receptor 5-HT3 receptor 5-HT5 receptor 5-HT6 receptor 5-HT7 receptor GRCh38: Ensembl release...
18 KB (2,073 words) - 06:23, 10 July 2024
Wesołowska A (2002). "In the search for selective ligands of 5-HT5, 5-HT6 and 5-HT7 serotonin receptors" (PDF). Polish Journal of Pharmacology. 54 (4): 327–341...
65 KB (5,263 words) - 10:40, 12 August 2024
5-hydroxytryptamine receptor 1B also known as the 5-HT1B receptor is a protein that in humans is encoded by the HTR1B gene. The 5-HT1B receptor is a 5-HT...
17 KB (1,982 words) - 06:24, 10 July 2024
pineal gland. 5-MT acts as a full agonist at the 5-HT1, 5-HT2, 5-HT4, 5-HT6, and 5-HT7 receptors. It has no affinity for the 5-HT3 receptor and its affinity...
7 KB (622 words) - 18:32, 11 August 2024
cognition and memory. AS-19 is a 5-HT7 receptor agonist that has been used in scientific research. Serotonin receptor antagonist "Eltoprazine - Elto Pharma...
16 KB (1,657 words) - 17:23, 8 June 2024
5-hydroxytryptamine (serotonin) receptor 1D, also known as HTR1D, is a 5-HT receptor, but also denotes the human gene encoding it. 5-HT1D acts on the central...
11 KB (1,237 words) - 06:53, 10 July 2024
The 5-HT2C receptor is a subtype of the 5-HT2 receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5-HT). Like all 5-HT2...
51 KB (6,098 words) - 04:17, 12 August 2024
Buspirone (category 5-HT1A agonists)
the serotonin 5-HT2A, 5-HT2B, 5-HT2C, 5-HT6, 5-HT7 receptors probably as an antagonist. In addition to binding to serotonin receptors, buspirone is an...
42 KB (3,631 words) - 13:44, 27 July 2024
The 5HT6 receptor is a subtype of 5HT receptor that binds the endogenous neurotransmitter serotonin (5-hydroxytryptamine, 5HT). It is a G protein-coupled...
29 KB (3,301 words) - 21:37, 9 March 2024
high-affinity full agonist at the 5-HT1A, 5-HT1B, 5-HT1D, 5-HT5A, and 5-HT7 receptors, as well as at the 5-HT2, 5-HT3, 5-HT6 receptors with lower affinity. It has...
6 KB (518 words) - 17:39, 12 August 2023
Serotonin modulator and stimulator (category Serotonin receptor antagonists)
serotonin reuptake inhibitor (SRI), agonist of the 5-HT1A receptor, and antagonist of the 5-HT3 and 5-HT7 receptors. However, it can also technically be applied...
5 KB (568 words) - 17:03, 21 March 2024
Brexpiprazole (category 5-HT7 antagonists)
release that is triggered by 5-HT1A receptor agonism. It is also an antagonist of the serotonin 5-HT2A, 5-HT2B, and 5-HT7 receptors, which may contribute to...
31 KB (2,342 words) - 16:44, 31 July 2024
The 5-HT3 antagonists, informally known as "setrons", are a class of drugs that act as receptor antagonists at the 5-HT3 receptor, a subtype of serotonin...
43 KB (4,628 words) - 10:52, 21 February 2024
Aripiprazole (category 5-HT7 antagonists)
that could be low (5-HT2A, 5-HT7), intermediate (D2L, 5-HT1A), or high (5-HT2C). This mixture of agonist actions at D2-dopamine receptors is consistent with...
105 KB (9,710 words) - 19:54, 1 August 2024
Muscarinic antagonist (redirect from Muscarinic receptor antagonists)
Huang XP, Tran TB, Meltzer HY, Roth BL (2009). "Amisulpride is a potent 5-HT7 antagonist: relevance for antidepressant actions in vivo". Psychopharmacology...
40 KB (1,998 words) - 10:32, 22 May 2024
δ1, δ2, κ Serotonergic: 5-HT1A, 5-HT1B, 5-HT1D, 5-HT1E, 5-HT1F, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT3, 5-HT4, 5-HT5, 5-HT6, 5-HT7 Autoreceptor Catecholamines...
16 KB (1,590 words) - 01:49, 26 October 2023
5-Hydroxytryptamine receptor 2B (5-HT2B) also known as serotonin receptor 2B is a protein that in humans is encoded by the HTR2B gene. 5-HT2B is a member...
32 KB (3,496 words) - 05:38, 10 July 2024
5-HT5B receptor is a 5-HT receptor protein and the gene which encodes it. The protein is found in rodents, but not in humans, because stop codons in the...
3 KB (348 words) - 07:25, 24 December 2023
8-OH-DPAT (category 5-HT7 agonists)
Originally believed to be selective for the 5-HT1A receptor, 8-OH-DPAT was later found to act as a 5-HT7 receptor agonist and serotonin reuptake inhibitor/releasing...
10 KB (875 words) - 21:03, 10 March 2024
rats using this compound while characterizing various agonists of the 5-HT7 receptor. It is an agonist with a Ki value of 630.96nM. Very little other data...
4 KB (295 words) - 19:40, 13 August 2023
5-HT1F (HTR1F, 5H1F) 5-HT4 (HTR4) InterPro: IPR001520 5-HT5A (HTR5A, 5H5A) 5-HT7 (HTR7, 5H7) InterPro: IPR001069 Olfactory receptor InterPro: IPR000725...
25 KB (2,172 words) - 01:01, 29 November 2023
Myenteric plexus (section Receptors)
; Heredia, D. J.; Smith, T. K. (2010). "Critical role of 5-HT1A, 5-HT3, and 5-HT7 receptor subtypes in the initiation, generation, and propagation of...
12 KB (1,431 words) - 09:16, 6 July 2024
Clomipramine (category Serotonin receptor antagonists)
α1-adrenergic receptor, the histamine H1 receptor, the serotonin 5-HT2A, 5-HT2C, 5-HT3, 5-HT6, and 5-HT7 receptors, the dopamine D1, D2, and D3 receptors, and...
117 KB (11,679 words) - 11:40, 24 July 2024