A prodrug is a pharmacologically inactive medication or compound that, after intake, is metabolized (i.e., converted within the body) into a pharmacologically...

Directed enzyme prodrug therapy (DEPT) uses enzymes artificially introduced into the body to convert prodrugs, which have no or poor biologically activity...

(γ-hydroxybutyric acid acetate) – synthetic prodrug to GHB GBL (γ-hydroxybutyric acid lactone) – metabolic intermediate and prodrug to GHB GHBAL (γ-hydroxybutyraldehyde...

estrogen in such research. However, NETE, an intramuscularly administered prodrug of norethisterone which is used as a long-acting contraceptive, is used...

Hypoxia-Activated Prodrugs (HAPs) are prodrugs that target regions of tumor hypoxia within tumor cells. HAPs may offer the potential, alone and in combination...

of mometasone, is the marketed medication. Mometasone furoate acts as a prodrug of mometasone. In addition to its glucocorticoid activity, mometasone also...

psilocybin for pharmacological studies, as they are both believed to be prodrugs of psilocin. However, some users report that O-acetylpsilocin's subjective...

Corticosteroids are a class of steroid hormones that are produced in the adrenal cortex of vertebrates, as well as the synthetic analogues of these hormones...

damage. Boldenone undecylenate is an androgen ester and a long-lasting prodrug of boldenone in the body. Boldenone undecylenate was introduced for medical...

called prodrugs. The reasons for this type of formulation may be because the drug is more stable during manufacture and storage as the prodrug form, or...

research chemical by online retailers. Due to its similarity to the psilocin prodrug 4-AcO-DMT, which is deacetylated to form psilocin in vivo, it is expected...

modulators mAChRsTooltip Muscarinic acetylcholine receptors Precursors (and prodrugs) Acetyl-coA Adafenoxate Choline (lecithin) Citicoline Cyprodenate Dimethylethanolamine...

L-threo-DOPS and SM-5688) is a synthetic amino acid precursor which acts as a prodrug to the neurotransmitter norepinephrine (noradrenaline). Unlike norepinephrine...

Levomethorphan is a prodrug to levorphanol, analogously to DXM acting as a prodrug to dextrorphan or codeine behaving as a prodrug to morphine. As such...

an androgen and testosterone prodrug Δ1-Androstenediol (Δ1-androsten-3β,17β-diol) – an androgen and δ1-testosterone prodrug Androstenedione Δ4-Androstenedione...

the lysine-analog of enalapril. Unlike other ACE inhibitors, it is not a prodrug, is not metabolized by the liver, and is excreted unchanged in the urine...

bacterium Moraxella catarrhalis. Tributyrin is a stable and rapidly absorbed prodrug of butyric acid which enhances antiproliferative effects of dihydroxycholecalciferol...

chemical that has potential psychedelic effects. It is believed to be a prodrug for LSD and has replaced 1V-LSD in Germany after 1V-LSD became covered...

is not recommended by the manufacturer. Lisdexamfetamine is an inactive prodrug that works after being converted by the body into dextroamphetamine, a...

received regulatory approval in 1991. Nabumetone is a non-acidic NSAID prodrug that is rapidly metabolized in the liver to the active metabolite, 6-methoxy-2-naphthyl...

dipropionate is the USAN and former BAN. It is a prodrug of the free form, beclometasone (INN). The prodrug beclometasone is marketed in Norway and Russia...

His main research focus has been on the design and characterization of prodrugs and protoxins targeted for activation by cancer specific proteases. This...

medicine used to treat (chronic) infections with hepatitis B virus. A prodrug form of adefovir was previously called bis-POM PMEA, with trade names Preveon...

cause these actions either separately or in combination. A variety of prodrugs of amphetamine and/or methamphetamine exist, and include amfecloral, amphetaminil...

calcitriol, via injection, may improve treatment outcomes. Paracetamol ester prodrug containing L-pyroglutamic acid (PGA), a biosynthetic precursor of glutathione...

liver damage worse in a dose-dependent fashion. Acetylcysteine serves as a prodrug to L-cysteine, a precursor to the biologic antioxidant glutathione. Hence...

olmesartan, the metabolism of the drug is unusual as it is a cascading prodrug. Candesartan has good bioavailibility and is the most potent by weight...

an anticonvulsant and analgesic drug of the gabapentinoid class, and a prodrug to gabapentin. It was designed for increased oral bioavailability over...

used for the treatment of Parkinson's disease. It is a combination of prodrugs for levodopa and carbidopa that is developed by AbbVie The combination...

substituted amphetamine derivative with empathogenic effects, which acts as a prodrug for MDA with a slower onset of effects and longer duration of action. Lys-MDA...